SCHEMBL6563671

SCHEMBL6563671

O=C(O)CNC(=O)Oc1nc2ccccc2cc1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 2/20 0.48
EGLN1 Q9GZT9 9/20 0.40
KDM4E B2RXH2 5/20 0.40
ALDH1A1 P00352 4/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 3/20 0.40
HPGD P15428 1/20 0.40
STAT3 P40763 1/20 0.40
FTO Q9C0B1 7/20 0.39
EGLN3 Q9H6Z9 2/20 0.39
KDM5B Q9UGL1 2/20 0.39
KDM2A Q9Y2K7 2/20 0.39
HIF1AN Q9NWT6 1/20 0.39
KDM6B O15054 2/20 0.38
PRNP P04156 2/20 0.38
RXFP1 Q9HBX9 2/20 0.38
EGLN2 Q96KS0 1/20 0.37
BBOX1 O75936 1/20 0.36
KDM3A Q9Y4C1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2549260 0.83 EGLN1 (0.39) EGLN1EGLN3HIF1ANRXFP1BBOX1
SCHEMBL8785457 0.83 KDM4C (0.45) KDM4CKDM4EALDH1A1MEN1KMT2A
SCHEMBL6564086 0.79 ALDH1A1 (0.49) KDM4EALDH1A1MEN1KMT2AGAA
SCHEMBL6567209 0.76 KDM4C (0.58) KDM4CEGLN1KDM4EALDH1A1MEN1
SCHEMBL821712 0.76 KDM4C (0.58) KDM4CEGLN1KDM4EALDH1A1MEN1
SCHEMBL8784892 0.73 TLR8 (0.43) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL6567506 0.72 ALDH1A1 (0.49) KDM4EALDH1A1MEN1KMT2AGAA
SCHEMBL4070937 0.71 FTO (0.57) EGLN1ALDH1A1GAAFTOEGLN3
SCHEMBL4076740 0.69 EGLN1 (0.44) KDM4CEGLN1KDM4EALDH1A1MEN1
SCHEMBL8779261 0.69 EGLN1 (0.38) EGLN1FTOEGLN3EGLN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0765871-B1 Substituted Quinoline-2-carboxamides, their preparation and their use as prolyle-4-hydroxylase Inhibitors FIBROGEN INC (US) 2004-03-31 EP disclosed
EP-0765871-A1 Substituted Quinoline-2-carboxamides, their preparation and their use as prolyle-4-hydroxylase Inhibitors HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-02 EP disclosed
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed