SCHEMBL6571774

SCHEMBL6571774

O=C([O-])CCSC1c2ccccc2C=Cc2ccc(OCc3ccc4cc(F)c(Cl)cc4n3)cc21.[Na+]

nearest known ligand 0.42

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALOX5AP known ✓ P20292 6/20 0.35
CYSLTR1 known ✓ Q9Y271 5/20 0.34
CYSLTR2 Q9NS75 4/20 0.34
TBXA2R P21731 1/20 0.34
GPBAR1 Q8TDU6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5335837 0.92 CYSLTR1 (0.39) ALOX5APCYSLTR1CYSLTR2TBXA2RGPBAR1
SCHEMBL4056757 0.84 CYSLTR2 (0.37) ALOX5APCYSLTR1CYSLTR2
SCHEMBL5333781 0.81 PDE10A (0.40) ALOX5APCYSLTR1CYSLTR2GPBAR1
SCHEMBL5333732 0.80 CYSLTR1 (0.45) CYSLTR1CYSLTR2TBXA2R
SCHEMBL5333735 0.80 CYSLTR1 (0.45) CYSLTR1CYSLTR2TBXA2R
SCHEMBL4053392 0.77 CYSLTR1 (0.39) ALOX5APCYSLTR1CYSLTR2GPBAR1
SCHEMBL5331476 0.77 TBXA2R (0.42) TBXA2R
SCHEMBL4052136 0.74 CYSLTR2 (0.36) ALOX5APCYSLTR1CYSLTR2
SCHEMBL5339124 0.74 CYSLTR1 (0.45) CYSLTR1CYSLTR2
SCHEMBL5339118 0.74 CYSLTR1 (0.45) CYSLTR1CYSLTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1408033-A1 DIBENZOCYCLOHEPTENE COMPOUND Ube Industries, Ltd. (JP) 2004-04-14 EP disclosed