SCHEMBL6572946

SCHEMBL6572946

COCCN(CCOC)c1ccc(N)c(-c2cccc(C(=O)O)c2)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 2/20 0.42
ATR Q13535 1/20 0.40
F2 P00734 1/20 0.40
PRSS1 P07477 1/20 0.40
PRSS2 P07478 1/20 0.40
PRSS3 P35030 1/20 0.40
PTGER4 P35408 1/20 0.40
KMO O15229 1/20 0.38
NR1H4 Q96RI1 2/20 0.38
PTGER1 P34995 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
FNTA P49354 1/20 0.38
FNTB P49356 1/20 0.38
PGGT1B P53609 1/20 0.38
FOLH1 Q04609 1/20 0.38
PLA2G2A P14555 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6574651 0.94 LMNA (0.43) PTPN11ATRF2PRSS1PRSS2
SCHEMBL6574647 0.93 PTGER1 (0.45) PTPN11ATRF2PRSS1PRSS2
SCHEMBL6572668 0.87 RARB (0.43) PTPN11F2PRSS1PRSS2PRSS3
SCHEMBL6573465 0.85 KMO (0.42) PTPN11KMOPTGER1AKR1C3AKR1C2
SCHEMBL6574642 0.85 LTB4R2 (0.43) PTPN11F2PRSS1PRSS2PRSS3
SCHEMBL6571441 0.83 CYP3A4 (0.38) F2PRSS1PRSS2PRSS3
SCHEMBL6571371 0.83 MAOA (0.34) F2PRSS1PRSS2PRSS3
SCHEMBL6572821 0.82 ALDH1A1 (0.37)
SCHEMBL6574166 0.82 MAP4K4 (0.42)
SCHEMBL6572734 0.81 FYN (0.44) ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed