SCHEMBL659126

SCHEMBL659126

Brc1cccc2ncsc12

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MAPK9 P45984 1/20 0.37
BACE1 P56817 1/20 0.34
PSMB8 P28062 1/20 0.33
PDPK1 O15530 1/20 0.33
CCKBR P32239 1/20 0.33
EGFR P00533 2/20 0.31
PRMT5 O14744 1/20 0.31
OPRM1 P35372 1/20 0.30
OPRL1 P41146 1/20 0.30
GRM5 P41594 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30081471 0.74 ALDH1A1 (0.45) ALDH1A1HSD17B10OPRM1OPRL1
SCHEMBL928489 0.74 ALDH1A1 (0.45) ALDH1A1HSD17B10MAPK9PSMB8PRMT5
SCHEMBL115601 0.74 ALDH1A1 (0.45) ALDH1A1HSD17B10OPRM1OPRL1
SCHEMBL2093035 0.74 ALDH1A1 (0.45) ALDH1A1HSD17B10MAPK9EGFRPRMT5
SCHEMBL115602 0.74 ALDH1A1 (0.45) ALDH1A1HSD17B10PRMT5OPRM1OPRL1
SCHEMBL5562354 0.74 ALDH1A1 (0.45) ALDH1A1HSD17B10CCKBRPRMT5OPRM1
SCHEMBL6972765 0.74 ALDH1A1 (0.45) ALDH1A1HSD17B10PRMT5OPRM1OPRL1
SCHEMBL288616 0.74 ALDH1A1 (0.45) ALDH1A1HSD17B10PRMT5OPRM1OPRL1
SCHEMBL9853741 0.74 ALDH1A1 (0.45) ALDH1A1HSD17B10PRMT5OPRM1OPRL1
SCHEMBL29806829 0.74 ALDH1A1 (0.45) ALDH1A1HSD17B10MAPK9EGFRPRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 156 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110098292-A1 New Compounds Useful for Treating CNS Disorders ASTRAZENECA AB (SE) 2011-04-28 US claimed
CN-1980922-A New compounds useful for treating CNS disorders ASTRAZENECA AB (SE) 2007-06-13 CN claimed
EP-1765815-A2 NEW COMPOUNDS USEFUL FOR TREATING CNS DISORDERS AstraZeneca AB (SE) 2007-03-28 EP claimed
WO-2006004507-A2 NEW BENZOTHIAZOLE DERIVATIVES USEFUL FOR TREATING CNS DISORDERS ASTRAZENECA AB (SE) 2006-01-12 WO claimed
US-12637449-B2 Organic compound and organic light emitting device including the same LG DISPLAY CO., LTD. (KR) 2026-05-26 US disclosed
US-20260103471-A1 CYCLIC UREA THIAZOLYL COMPOUNDS FOR TREATMENT OF HSV ASSEMBLY BIOSCIENCES INC (US) 2026-04-16 US disclosed
US-20260014146-A1 CDK2 INHIBITORS AND METHODS OF USING THE SAME CEDILLA THERAPEUTICS INC (US) 2026-01-15 US disclosed
US-20250376478-A1 CYCLIC UREA THIAZOLYL COMPOUNDS FOR TREATMENT OF HSV ASSEMBLY BIOSCIENCES INC (US) 2025-12-11 US disclosed
US-12478621-B2 Substituted aminoquinolones as dgkalpha inhibitors for immune activation DEUTSCHES KREBSFORSCHUNGSZENTRUM (DE) 2025-11-25 US disclosed
US-20250270215-A1 IMIDAZOLE DERIVATIVES AS ALK5 INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2025-08-28 US disclosed
EP-4581029-A1 CYCLIC UREA THIAZOLYL COMPOUNDS FOR TREATMENT OF HSV Assembly Biosciences, Inc. (US) 2025-07-09 EP disclosed
EP-4562014-A2 CDK2 INHIBITORS AND METHODS OF USING THE SAME Cedilla Therapeutics, Inc. (US) 2025-06-04 EP disclosed
EP-2393806-A1 INHIBITORS OF JUN N-TERMINAL KINASE Elan Pharmaceuticals Inc. (US) 2011-12-14 EP disclosed
WO-2011100502-A1 7-AMINOFUROPYRIDINE DERIVATIVES OSI Pharmaceuticals, LLC (US) 2011-08-18 WO disclosed
US-20110098292-A1 New Compounds Useful for Treating CNS Disorders ASTRAZENECA AB (SE) 2011-04-28 US disclosed
US-20100331335-A1 Inhibitors of Jun N-Terminal Kinase ELAN PHARMACETICALS, INC. 2010-12-30 US disclosed
WO-2010091310-A1 INHIBITORS OF JUN N-TERMINAL KINASE ELAN PHARMACEUTICALS, INC. (US) 2010-08-12 WO disclosed
CN-1980922-A New compounds useful for treating CNS disorders ASTRAZENECA AB (SE) 2007-06-13 CN disclosed
EP-1765815-A2 NEW COMPOUNDS USEFUL FOR TREATING CNS DISORDERS AstraZeneca AB (SE) 2007-03-28 EP disclosed
WO-2006004507-A2 NEW BENZOTHIAZOLE DERIVATIVES USEFUL FOR TREATING CNS DISORDERS ASTRAZENECA AB (SE) 2006-01-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260103471-A1 CYCLIC UREA THIAZOLYL COMPOUNDS FOR TREATMENT OF HSV TK1, UNG, SMCHD1 ALDH1A1 3205/4885HSD17B10 2667/4885MAPK9 1204/4885
US-12478621-B2 Substituted aminoquinolones as dgkalpha inhibitors for immune activation DGKK, DGKG, DGKA ALDH1A1 3915/4885HSD17B10 3531/4885MAPK9 416/4885
US-12637449-B2 Organic compound and organic light emitting device including the same CRY1, NR2E3, CRY2 ALDH1A1 289/4885HSD17B10 875/4885MAPK9 4313/4885
US-20110098292-A1 New Compounds Useful for Treating CNS Disorders SLC18A2, PMP22, GAP43 ALDH1A1 1045/4885HSD17B10 1386/4885MAPK9 3486/4885
US-20250376478-A1 CYCLIC UREA THIAZOLYL COMPOUNDS FOR TREATMENT OF HSV TYMP, TK1, TREH ALDH1A1 3189/4885HSD17B10 3385/4885MAPK9 2410/4885
US-20250270215-A1 IMIDAZOLE DERIVATIVES AS ALK5 INHIBITORS ALK, TGFBR1, TGFBR2 ALDH1A1 828/4885HSD17B10 3765/4885MAPK9 410/4885
US-20100331335-A1 Inhibitors of Jun N-Terminal Kinase CHUK, MAPK6, MAPK3 ALDH1A1 4529/4885HSD17B10 3960/4885MAPK9 16/4885
US-20260014146-A1 CDK2 INHIBITORS AND METHODS OF USING THE SAME CDK2, CDK20, CDK1 ALDH1A1 3585/4885HSD17B10 1442/4885MAPK9 718/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.