SCHEMBL6609399

SCHEMBL6609399

Cc1cccc(N2CC(OC(=O)Nc3ccc(N(C)c4nc(C)cc(C)n4)cc3)CC2=O)c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.41
GAA P10253 3/20 0.41
MAPT P10636 5/20 0.41
HPGD P15428 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MCL1 Q07820 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HIF1A Q16665 1/20 0.41
HSD17B10 Q99714 2/20 0.40
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
LMNA P02545 1/20 0.36
USP2 O75604 1/20 0.36
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6611399 0.89 ALDH1A1 (0.41) ALDH1A1GAAMAPTHPGDNPSR1
SCHEMBL6613841 0.86 ALDH1A1 (0.39) ALDH1A1MAPTHPGDNPSR1KDM4E
SCHEMBL6611945 0.86 ALDH1A1 (0.47) ALDH1A1GAAMAPTHPGDKDM4E
SCHEMBL5842523 0.85 ALDH1A1 (0.58) ALDH1A1GAAMAPTHPGDNPSR1
SCHEMBL6609900 0.82 ALOX15 (0.43) ALDH1A1MAPTHPGDNPSR1KDM4E
SCHEMBL6613611 0.82 ACHE (0.42) ALDH1A1MAPTHPGDNPSR1KDM4E
SCHEMBL6611922 0.81 ALDH1A1 (0.48) ALDH1A1MAPTHPGDNPSR1KDM4E
SCHEMBL6611410 0.81 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL6615359 0.81 MAPT (0.39) ALDH1A1MAPTHPGDNPSR1KDM4E
SCHEMBL6614115 0.79 ALDH1A1 (0.49) ALDH1A1MAPTSMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1463724-A1 PYRROLIDONE CARBOXAMIDES Actelion Pharmaceuticals Ltd. (CH) 2004-10-06 EP disclosed
WO-2003059905-A1 PYRROLIDONE CARBOXAMIDES ACTELION PHARMACEUTICALS LTD (CH) 2003-07-24 WO disclosed