SCHEMBL662265

SCHEMBL662265

COc1c(C)c(O)c(C)c(O)c1C(=O)/C=C/c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 1.00
KCNA3 P22001 5/20 0.59
MAPT P10636 5/20 0.58
NPSR1 Q6W5P4 3/20 0.58
MAOB P27338 2/20 0.57
CYP19A1 P11511 1/20 0.57
CYP2C9 P11712 1/20 0.57
MAOA P21397 1/20 0.57
CYP2C19 P33261 1/20 0.57
TNFRSF1A P19438 3/20 0.53
KMT2A Q03164 3/20 0.53
MEN1 O00255 2/20 0.53
TP53 P04637 1/20 0.52
CYP3A4 P08684 1/20 0.52
ATM Q13315 1/20 0.52
HSD17B10 Q99714 1/20 0.52
CYP1B1 Q16678 3/20 0.50
CYP1A1 P04798 2/20 0.50
ALDH1A1 P00352 1/20 0.50
HSPD1 P10809 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL662266 1.00 ABCB1 (1.00) ABCB1KCNA3MAPTNPSR1MAOB
SCHEMBL25340278 0.89 ABCB1 (0.80) ABCB1KCNA3MAPTMAOBMAOA
SCHEMBL662284 0.89 ABCB1 (0.80) ABCB1KCNA3MAPTMAOBMAOA
SCHEMBL662283 0.89 ABCB1 (0.80) ABCB1KCNA3MAPTMAOBMAOA
SCHEMBL25952345 0.89 ABCB1 (0.80) ABCB1KCNA3MAPTMAOBMAOA
SCHEMBL25337768 0.88 ABCB1 (0.78) ABCB1MAPTMAOBCYP2C9MAOA
SCHEMBL25952365 0.88 ABCB1 (0.78) ABCB1MAPTMAOBCYP2C9MAOA
SCHEMBL25340515 0.86 ABCB1 (0.76) ABCB1KCNA3MAPTMAOBMAOA
SCHEMBL25340711 0.86 ABCB1 (0.76) ABCB1KCNA3MAPTMAOBMAOA
SCHEMBL25952337 0.86 ABCB1 (0.76) ABCB1KCNA3MAPTMAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023177191-A1 COMPOSITION FOR PREVENTING OR TREATING FIBROTIC DISEASES, COMPRISING DIMETHYLCHALCONE DERIVATIVE AS ACTIVE INGREDIENT 서울대학교 산학협력단 2023-09-21 WO claimed
US-20230248665-A1 COMPOSITION COMPRISING DIMETHYLCHALCONE DERIVATIVE FOR PREVENTION OR TREATMENT OF METABOLIC DISEASE SEOUL NATIONAL UNIVERSITY R & DB FOUNDATION (KR) 2023-08-10 US claimed
US-20120046353-A1 CLEISTOCALYX OPERCULATUS-DERIVED COMPOUNDS HAVING INHIBITORY ACTIVITIES AGAINST AVIAN AND SWINE INFLUENZA VIRUSES OR NOVEL INFLUENZA VIRUS CHOONG ANG VACCINE LAB. (KR) 2012-02-23 US claimed
WO-2012023660-A1 ANTIVIRAL DRUG FOR AVIAN AND SWINE INFLUENZA AND NOVEL FLU, OBTAINED FROM CLEISTOCALYX OPERCULATUS 주식회사 중앙백신연구소 (KR) 2012-02-23 WO claimed
US-12428405-B2 Chalcone-based chemotherapeutic compound for triple negative breast cancer QATAR UNIVERSITY (QA) 2025-09-30 US disclosed
WO-2024189607-A1 METHODS AND BIOAVAILABLE HIGHLY PERMEABLE COMPOUNDS FOR DISEASES TREATMENT DIDENKO KIRILL (MX) 2024-09-19 WO disclosed
US-20230365539-A1 NOVEL CHALCONE-BASED CHEMOTHERAPEUTIC COMPOUND FOR TRIPLE NEGATIVE BREAST CANCER QATAR UNIVERSITY (QA) 2023-11-16 US disclosed
US-20230295103-A1 AURONE DERIVATIVES AND USES THEREOF FOR CONTROLLING BACTERIA AND/OR FUNGI ECOLE CENTRALE DE MARSEILLE (FR) 2023-09-21 US disclosed
WO-2023177191-A1 COMPOSITION FOR PREVENTING OR TREATING FIBROTIC DISEASES, COMPRISING DIMETHYLCHALCONE DERIVATIVE AS ACTIVE INGREDIENT 서울대학교 산학협력단 2023-09-21 WO disclosed
WO-2023177191-A1 COMPOSITION FOR PREVENTING OR TREATING FIBROTIC DISEASES, COMPRISING DIMETHYLCHALCONE DERIVATIVE AS ACTIVE INGREDIENT 서울대학교 산학협력단 2023-09-21 WO disclosed
WO-2023177194-A1 NOVEL DIMETHYLCHALCONE DERIVATIVES 중앙대학교 산학협력단 2023-09-21 WO disclosed
WO-2023177194-A1 NOVEL DIMETHYLCHALCONE DERIVATIVES 중앙대학교 산학협력단 2023-09-21 WO disclosed
CN-101259118-A Application of 2',4'-dihydroxy-6'-methoxy-3',5'-dimethyl chalcone as PPAR gamma agonist GUANGZHOU INST BIOMED & HEALTH (CN) 2008-09-10 CN disclosed
US-20080166304-A1 Inactivation of Microorganisms With Multidrug Resistance Inhibitors and Phenothiaziniums THE GENERAL HOSPITAL CORPOARTION (US) 2008-07-10 US disclosed
CN-100357264-C Charles ketone oxime and its composition , preparation method and uses SOUTH CHINA BOTAN GARDEN CHINE (CN) 2007-12-26 CN disclosed
CN-1275923-C Use of 2',4'-dihydroxy-6'-methoxy-3',5'-dimethyl chalkone as reversing agent for resistance of multiple tumours drugs UNIV EAST CHINA SCIENCE & TECH (CN) 2006-09-20 CN disclosed
CN-1807405-A Charles ketone oxime and its composition , preparation method and uses SOUTH CHINA BOTAN GARDEN CHINE (CN) 2006-07-26 CN disclosed
CN-1680248-A Use of 2',4'-dihydroxy-6'-methoxy-3',5'-dimethyl chalkone as reversing agent for resistance of multiple tumours drugs HUADONG SCIENCE & ENGINEERING (CN) 2005-10-12 CN disclosed
CN-1680248-A Use of 2',4'-dihydroxy-6'-methoxy-3',5'-dimethyl chalkone as reversing agent for resistance of multiple tumours drugs HUADONG SCIENCE & ENGINEERING (CN) 2005-10-12 CN disclosed
CN-1454895-A Use of 2',4'-dihydroxy-6'-methoxy-3',5'-dimethyl chalcone for preparing anticancer medicine TUMOUR PREVENTION AND TREAT CT (CN) 2003-11-12 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120046353-A1 CLEISTOCALYX OPERCULATUS-DERIVED COMPOUNDS HAVING INHIBITORY ACTIVITIES AGAINST AVIAN AND SWINE INFLUENZA VIRUSES OR NOVEL INFLUENZA VIRUS PIGS, CLEC4M, ENGASE ABCB1 4746/4885KCNA3 2228/4885MAPT 2192/4885
US-12428405-B2 Chalcone-based chemotherapeutic compound for triple negative breast cancer BRCA1, TOP2B, TOP1 ABCB1 8/4885KCNA3 4339/4885MAPT 1698/4885
US-20230295103-A1 AURONE DERIVATIVES AND USES THEREOF FOR CONTROLLING BACTERIA AND/OR FUNGI AURKA, CYP51A1, AURKC ABCB1 1680/4885KCNA3 1929/4885MAPT 2614/4885
US-20230248665-A1 COMPOSITION COMPRISING DIMETHYLCHALCONE DERIVATIVE FOR PREVENTION OR TREATMENT OF METABOLIC DISEASE LIPC, PC, CYP27A1 ABCB1 3180/4885KCNA3 4014/4885MAPT 1563/4885
US-20230365539-A1 NOVEL CHALCONE-BASED CHEMOTHERAPEUTIC COMPOUND FOR TRIPLE NEGATIVE BREAST CANCER BRCA1, PGR, TOP2B ABCB1 21/4885KCNA3 4277/4885MAPT 2108/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.