SCHEMBL6631331

SCHEMBL6631331

[CH2]C(OCC)(OCC)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
ALOX15 P16050 1/20 0.41
KCNN4 O15554 2/20 0.40
MAPK1 P28482 1/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 2/20 0.38
KIF11 P52732 1/20 0.38
HIF1A Q16665 1/20 0.38
LMNA P02545 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
EDNRB P24530 1/20 0.36
EDNRA P25101 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ESR1 P03372 2/20 0.35
ESR2 Q92731 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
PIN1 Q13526 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27859509 0.86 LTA4H (0.37) ALDH1A1ALOX15KCNN4MAPK1CYP3A4
SCHEMBL27691475 0.83 ALDH1A1 (0.39) ALDH1A1ALOX15KCNN4MAPK1CYP3A4
SCHEMBL27801514 0.82 KCNN4 (0.40) ALDH1A1ALOX15KCNN4MAPK1CYP3A4
SCHEMBL27662558 0.78 MEN1 (0.45) MAPK1CYP3A4HIF1ALMNASMN1; SMN2
SCHEMBL27766103 0.78 KCNN4 (0.38) ALDH1A1ALOX15KCNN4MAPK1CYP3A4
SCHEMBL11355373 0.77 ALDH1A1 (0.41) ALDH1A1ALOX15KCNN4MAPK1CYP3A4
SCHEMBL3365376 0.77 POLB (0.41) ALDH1A1ALOX15KCNN4MAPK1CYP3A4
SCHEMBL27473812 0.77 SCN5A (0.41) ALDH1A1KIF11LMNAMAPT
SCHEMBL2350021 0.76 KIF11 (0.56) ALDH1A1ALOX15KCNN4MAPK1KIF11
SCHEMBL379267 0.76 KCNN4 (0.43) ALDH1A1ALOX15KCNN4MAPK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101029022-B Process for producing nitrogen-containing aromatic ring derivative EISAI R&D MAN CO LTD 2011-01-12 CN disclosed
CN-101029022-A Process for producing nitrogen-containing aromatic ring derivative EISAI R&D MAN CO LTD (JP) 2007-09-05 CN disclosed
CN-101024627-A Nitrogen-containing aromatic ring derivatives EISAI R&D MAN CO LTD (JP) 2007-08-29 CN disclosed
CN-1308310-C Nitrogen-containing aromatic ring derivatives EISAI CO LTD (JP) 2007-04-04 CN disclosed
CN-1500086-A Aminopiperidine derivatives 霍夫曼-拉罗奇有限公司 2004-05-26 CN disclosed
US-6737429-B2 TREATMENT OF HIV MEDIATED DISEASES. HOFFMANN-LA ROCHE INC. 2004-05-18 US disclosed
EP-1417202-A2 AMINOPIPERIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY F. HOFFMANN-LA ROCHE AG (CH) 2004-05-12 EP disclosed
CN-1440385-A Pyrrole derivatives for the treatment of AIDS HOFFMANN LA ROCHE (CH) 2003-09-03 CN disclosed
EP-1301481-A1 PYRROLE DERIVATIVES FOR TREATING AIDS F. HOFFMANN-LA ROCHE AG (CH) 2003-04-16 EP disclosed
US-20030069276-A1 Amino piperidine derivatives F.HOFFMANN-LA ROCHE AG (CH) 2003-04-10 US disclosed
WO-2002079186-A2 AMINOPIPERIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY F. HOFFMANN-LA ROCHE AG (CH) 2002-10-10 WO disclosed
US-20020032221-A1 Pyrrole derivatives ROCHE PRODUCTS LIMITED (GB) 2002-03-14 US disclosed
WO-2002002524-A1 PYRROLE DERIVATIVES FOR TREATING AIDS F. HOFFMANN-LA ROCHE AG (CH) 2002-01-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030069276-A1 Amino piperidine derivatives CCR5, CCR2, CXCR4 ALDH1A1 1935/4885ALOX15 3235/4885KCNN4 4207/4885
US-20020032221-A1 Pyrrole derivatives PYCR1, SARS1, MAVS ALDH1A1 2902/4885ALOX15 2101/4885KCNN4 4860/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.