SCHEMBL6675971

SCHEMBL6675971

CCN=C(N)Nc1cccc(CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 1/20 0.43
SCN5A Q14524 1/20 0.43
GPR35 Q9HC97 1/20 0.39
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2B Q13224 1/20 0.36
GRIN2C Q14957 1/20 0.36
GRIN3A Q8TCU5 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
REN P00797 1/20 0.35
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
PTGIR P43119 2/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
MAPK1 P28482 1/20 0.34
PDK1 Q15118 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6676767 0.89 CACNA1C (0.43) CACNA1CSCN5AGPR35GRIN2DGRIN3B
SCHEMBL6678098 0.85 GPR35 (0.39) GPR35RENMEN1KMT2AMAPK1
SCHEMBL7242006 0.81 GPR35 (0.38) GPR35RENNOS3NOS1NOS2
SCHEMBL6675968 0.80 GPR35 (0.39) CACNA1CSCN5AGPR35RENMEN1
SCHEMBL7242001 0.79 GPR35 (0.38) GPR35RENMEN1KMT2AMAPK1
SCHEMBL6678030 0.78 SIGMAR1 (0.44) CACNA1CSCN5AGRIN2DGRIN3BGRIN1
SCHEMBL6676278 0.78 REN (0.37) GPR35RENMEN1KMT2AMAPK1
SCHEMBL6675317 0.76 CACNA1C (0.49) CACNA1CSCN5AGPR35GRIN2DGRIN3B
SCHEMBL6678068 0.76 REN (0.36) RENGRM2
Hydrochloric Acid SCHEMBL6674250 0.75 CACNA1C (0.48) CACNA1CSCN5AGPR35GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed