SCHEMBL65299

SCHEMBL65299

CCOC(=O)C1C(c2ccc(OCCOc3c(Cl)cccc3Cl)cc2)CCN(C(=O)O)C1CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.35
TSHR P16473 2/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
KCNH2 Q12809 3/20 0.33
REN P00797 3/20 0.33
MAPT P10636 2/20 0.33
CYP3A4 P08684 2/20 0.33
GRM5 P41594 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
PKM P14618 1/20 0.33
KMT2A Q03164 1/20 0.33
P2RX7 Q99572 1/20 0.32
EGFR P00533 2/20 0.32
KDM4E B2RXH2 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
GPR119 Q8TDV5 1/20 0.32
ESR1 P03372 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65814 0.92 PPARG (0.39) LTA4HTSHRALDH1A1NPC1RAB9A
SCHEMBL64035 0.79 SLC6A2 (0.37) TSHRNPC1RAB9AL3MBTL1GRM5
SCHEMBL64234 0.75 L3MBTL1 (0.36) LTA4HL3MBTL1KCNH2RENMAPT
SCHEMBL66855 0.75 ELANE (0.38)
SCHEMBL64233 0.69 CHRM5 (0.35) LTA4HL3MBTL1MAPTCYP3A4KDM4E
SCHEMBL15951884 0.69 RIPK1 (0.36) HRH3
SCHEMBL64057 0.68 PPARG (0.39) LTA4HTSHRL3MBTL1MAPTEGFR
SCHEMBL78781 0.68 KDM4E (0.36) LTA4HL3MBTL1KDM4EESR1ESR2
SCHEMBL66293 0.67 PPM1B (0.32)
SCHEMBL556677 0.67 REN (0.41) KCNH2RENCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed