SCHEMBL6686236

SCHEMBL6686236

C[C@@H](C(=O)NCC(C(=O)NCCC1CNc2ccc(F)cc21)C1CCCCC1)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRM7 Q14831 2/20 0.38
TP53 P04637 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
TRPV1 Q8NER1 1/20 0.33
PYGL P06737 1/20 0.33
OPRL1 P41146 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6685697 0.95 TRPV1 (0.35) GRM7TRPV1
SCHEMBL6689424 0.93 TRPV1 (0.34) GRM7TRPV1PYGL
SCHEMBL6687531 0.93 TRPV1 (0.34) TSHRTRPV1PYGL
SCHEMBL6688201 0.90 FAAH (0.43) MEN1KMT2ATRPV1
SCHEMBL6686227 0.83 CTSS (0.40) TRPV1
SCHEMBL6690648 0.82 NMT2 (0.45) GRM7
SCHEMBL6686987 0.82 CTSL (0.42) MEN1KMT2APYGL
SCHEMBL6689091 0.81 CTSL (0.41) MEN1KMT2A
SCHEMBL6690788 0.80 CTSD (0.38) TDP1KMT2A
SCHEMBL6689089 0.79 KMT2A (0.42) TSHRMEN1KMT2ATRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084843-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed