SCHEMBL6689089

SCHEMBL6689089

CS(=O)(=O)Nc1ccc(C(=O)NCC(C(=O)NCCC2CNc3ccc(F)cc32)C2CCCCC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 1/20 0.42
HTR1A P08908 1/20 0.37
HTR1D P28221 1/20 0.37
HTR1F P30939 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TSHR P16473 1/20 0.37
EPHX2 P34913 4/20 0.36
NR1H4 Q96RI1 2/20 0.35
CTSL P07711 1/20 0.35
NTRK1 P04629 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
ADRB1 P08588 1/20 0.33
MMP13 P45452 1/20 0.33
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
S1PR1 P21453 1/20 0.33
NAMPT P43490 1/20 0.33
CTSS P25774 1/20 0.33
PPARG P37231 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6690788 0.86 CTSD (0.38) KMT2AALDH1A1EPHX2NAMPTCTSS
SCHEMBL6686227 0.85 CTSS (0.40) ALDH1A1CTSLTRPV1CTSSPKM
SCHEMBL6689428 0.84 MEN1 (0.41) KMT2AALDH1A1MEN1
SCHEMBL6686987 0.84 CTSL (0.42) KMT2AALDH1A1CTSLCTSSMEN1
SCHEMBL6689091 0.83 CTSL (0.41) KMT2AALDH1A1SMN1; SMN2CTSLCTSS
SCHEMBL6692878 0.81 MEN1 (0.39) KMT2APRMT5MEN1
SCHEMBL6690045 0.81 ALDH1A1 (0.51) KMT2AALDH1A1SMN1; SMN2TSHREPHX2
SCHEMBL6685697 0.80 TRPV1 (0.35) HTR1AHTR1DHTR1FCTSLTRPV1
SCHEMBL6686236 0.79 GRM7 (0.38) KMT2ATSHRTRPV1MEN1
SCHEMBL6689424 0.78 TRPV1 (0.34) TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084843-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed