SCHEMBL6746020

SCHEMBL6746020

CS(=O)(=O)c1c(F)cc(C2=CCC=C2c2cccc(OC(F)(F)F)c2)cc1F

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 8/20 0.39
GALR1 P47211 1/20 0.38
PIM1 P11309 2/20 0.37
PIM2 Q9P1W9 2/20 0.37
PTGES2 Q9H7Z7 2/20 0.36
CCNT1 O60563 1/20 0.36
CDK9 P50750 1/20 0.36
XDH P47989 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
SCN9A Q15858 1/20 0.35
KCNH2 Q12809 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.35
KAT6A Q92794 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6743255 0.86 KIF11 (0.44) DHODHGALR1SCN9A
SCHEMBL6747448 0.82 NR1H2 (0.37) DHODHGALR1PIM1PIM2PTGES2
SCHEMBL6749791 0.81 PTGS2 (0.40)
SCHEMBL6746349 0.81 PTGS2 (0.41)
SCHEMBL6747092 0.80 KIF11 (0.33)
SCHEMBL6746687 0.80 PTGS2 (0.39)
SCHEMBL6745114 0.80 SDHB (0.38) GALR1
SCHEMBL6745120 0.79 ACLY (0.35)
SCHEMBL6743237 0.79 PTGS2 (0.38)
SCHEMBL6746293 0.79 PTGS2 (0.38) GALR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6699884-B2 ANTIINFLAMMATORY CYCLOOXYGENASE INHIBITORS. PHARMACIA CORPORATION 2004-03-02 US claimed
US-6699884-B2 ANTIINFLAMMATORY CYCLOOXYGENASE INHIBITORS. PHARMACIA CORPORATION 2004-03-02 US disclosed