SCHEMBL679527

SCHEMBL679527

Fc1ccc(Oc2cc(Oc3ccc(Cl)c(C(F)(F)F)c3)ncn2)cc1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 12/20 0.49
BRAF P15056 3/20 0.47
RAF1 P04049 4/20 0.45
MAPK3 P27361 4/20 0.45
HTR2A P28223 1/20 0.43
SLC6A4 P31645 1/20 0.43
KCNH2 Q12809 1/20 0.43
PLA2G7 Q13093 1/20 0.43
KMO O15229 1/20 0.43
FLT1 P17948 1/20 0.42
FLT4 P35916 1/20 0.42
MAP2K7 O14733 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7885604 0.93 RAF1 (0.49) KDRBRAFRAF1MAPK3PLA2G7
SCHEMBL8773801 0.93 KDR (0.47) KDRBRAFRAF1MAPK3PLA2G7
SCHEMBL6938479 0.91 KDR (0.48) KDRBRAFHTR2ASLC6A4KCNH2
SCHEMBL7781852 0.87 KDR (0.48) KDRBRAFRAF1MAPK3HTR2A
SCHEMBL8773800 0.87 KDR (0.48) KDRBRAFRAF1MAPK3HTR2A
SCHEMBL7776445 0.87 RAF1 (0.46) KDRBRAFRAF1MAPK3PLA2G7
SCHEMBL8199428 0.86 KDR (0.44) KDRBRAFRAF1MAPK3HTR2A
SCHEMBL7791086 0.86 KDR (0.49) KDRBRAFRAF1MAPK3PLA2G7
SCHEMBL679617 0.85 RAF1 (0.45) KDRBRAFRAF1MAPK3PLA2G7
SCHEMBL3366738 0.85 EGFR (0.46) KDRBRAFRAF1HTR2ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100204167-A1 ACTIVE COMPOUND COMBINATIONS HAVING INSECTICIDAL AND ACARICIDAL PROPERTIES BAYER CROPSCIENCE AG (DE) 2010-08-12 US claimed
EP-0883991-B1 Methods for improving the residual control of mites and prolonging the protection of plants from mite infestations BASF AG (DE) 2003-01-02 EP claimed
US-5883104-A APPLYING TO THE FOLIAGE OF PLANTS AN UNSYMMETRICAL 4,6-BIS(ARYLOXY)PYRIMIDINE COMPOUND AMERICAN CYANAMID COMPANY (US) 1999-03-16 US claimed
EP-0883991-A1 Methods for improving the residual control of mites and prolonging the protection of plants from mite infestations American Cyanamid Company (US) 1998-12-16 EP claimed
US-5707995-A APPLYING TO SKINS/COATS OF ANIMALS TO CONTROL TICKS, INSECTS, PARASITES AMERICAN CYANAMID COMPANY (US) 1998-01-13 US claimed
JP-11228311-A None JP disclosed
US-9173394-B2 Active agent combinations having insecticidal and acaricidal properties BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-11-03 US disclosed
US-8962672-B2 Active agent combinations with insecticidal and acaricidal properties BAYER CROPSCIENCE AG (DE) 2015-02-24 US disclosed
EP-1982594-B1 Active agent combinations with insecticidal and acaricidal properties BAYER CROPSCIENCE AG (DE) 2014-05-14 EP disclosed
US-8299036-B2 Active agent combinations with insecticidal and acaricidal properties BAYER CROPSCIENCE AG (DE) 2012-10-30 US disclosed
US-20120010076-A1 ACTIVE AGENT COMBINATIONS WITH INSECTICIDAL AND ACARICIDAL PROPERITIES BAYER CROPSCIENCE AG (DE) 2012-01-12 US disclosed
US-8044085-B2 Active agent combinations with insecticidal and acaricidal properties BAYER CROPSCIENCE AG (DE) 2011-10-25 US disclosed
US-6087498-A Process for the preparation of unsymmetrical 4,6-bis(aryloxy) pyrimidine compounds AMERICAN CYANAMID COMPANY (US) 2000-07-11 US disclosed
US-5977363-A Process for the preparation of unsymmetrical 4,6-bis(aryloxy) pyrimidine compounds AMERICAN CYANAMID COMPANY (US) 1999-11-02 US disclosed
JP-H11228311-A IMPROVEMENT OF RESIDUAL PREVENTION OF MITE AND METHOD FOR KEEPING PLANT PROTECTION FROM PARATISM OF THE SAME AMERICAN CYANAMID CO 1999-08-24 JP disclosed
EP-0902020-A1 Improved process for the preparation of unsymmetrical 4,6-bis (aryloxy) pyrimidine compounds American Cyanamid Company (US) 1999-03-17 EP disclosed
US-5883104-A APPLYING TO THE FOLIAGE OF PLANTS AN UNSYMMETRICAL 4,6-BIS(ARYLOXY)PYRIMIDINE COMPOUND AMERICAN CYANAMID COMPANY (US) 1999-03-16 US disclosed
EP-0883991-A1 Methods for improving the residual control of mites and prolonging the protection of plants from mite infestations American Cyanamid Company (US) 1998-12-16 EP disclosed
US-5849910-A Process for the preparation of unsymmetrical 4,6-bis aryloxy-pyrimidine compounds AMERICAN CYANAMID COMPANY (US) 1998-12-15 US disclosed
EP-0794177-A1 Process for the preparation of unsymmertical 4,6-Bis (aryloxy pyrimidine compounds American Cyanamid Company (US) 1997-09-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010076-A1 ACTIVE AGENT COMBINATIONS WITH INSECTICIDAL AND ACARICIDAL PROPERITIES ACAA2, ACHE, AADAC KDR 4766/4885BRAF 4084/4885RAF1 3027/4885
US-20100204167-A1 ACTIVE COMPOUND COMBINATIONS HAVING INSECTICIDAL AND ACARICIDAL PROPERTIES ACHE, ACAT2, ACAT1 KDR 4834/4885BRAF 4663/4885RAF1 4283/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.