SCHEMBL6814142

SCHEMBL6814142

COc1cc(C(N)=O)ccn1.Cc1c(=O)c(Cc2ccc(F)c(F)c2)cn2cc(C(=O)O)sc12

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 6/20 0.35
KDM5B Q9UGL1 6/20 0.35
TRPA1 O75762 1/20 0.35
KDM4C Q9H3R0 5/20 0.35
FYN P06241 1/20 0.34
STING1 Q86WV6 1/20 0.34
GRM2 Q14416 1/20 0.33
P2RX3 P56373 3/20 0.32
SCD O00767 1/20 0.32
GPR52 Q9Y2T5 1/20 0.31
MAPT P10636 1/20 0.31
P2RY14 Q15391 1/20 0.31
OPRK1 P41145 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6814148 0.90 LOXL2 (0.40) KDM5AKDM5BTRPA1KDM4CGRM2
SCHEMBL6819189 0.85 KDM5A (0.37) KDM5AKDM5BKDM4CFYNSTING1
SCHEMBL6484565 0.84 RXRA (0.35) KDM5AKDM5BTRPA1SCDMAPT
SCHEMBL6814145 0.82 TRPA1 (0.52) TRPA1SCDMAPT
SCHEMBL6819195 0.75 LOXL2 (0.40) KDM5AKDM5BTRPA1KDM4CGRM2
SCHEMBL6476858 0.71 TRPA1 (0.49) TRPA1MAPT
SCHEMBL6819192 0.70 MMP13 (0.41) TRPA1SCD
SCHEMBL6485426 0.69 P2RY14 (0.36) KDM5AKDM5BFYNSCDP2RY14
Niacinamide SCHEMBL6818598 0.69 FYN (0.39) FYNMAPTP2RY14
SCHEMBL6476888 0.66 RXRA (0.35) KDM5AKDM5BKDM4CP2RY14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014908-A1 HETEROBICYLCIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed