SCHEMBL6819192

SCHEMBL6819192

COc1cc(CNC(=O)c2cn3cc(Cc4ccc(F)c(F)c4)c(=O)c(C)c3o2)ccn1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 2/20 0.41
TRPA1 O75762 1/20 0.40
EPHX2 P34913 5/20 0.40
PDE10A Q9Y233 2/20 0.39
CDK2 P24941 1/20 0.37
GSK3B P49841 1/20 0.37
WDR5 P61964 2/20 0.37
PPARG P37231 1/20 0.36
SCD O00767 1/20 0.36
MET P08581 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
KLKB1 P03952 1/20 0.35
MAPK1 P28482 1/20 0.35
NTRK1 P04629 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6477930 0.88 MMP13 (0.48) MMP13TRPA1EPHX2CDK2GSK3B
SCHEMBL6819195 0.85 LOXL2 (0.40) MMP13TRPA1
SCHEMBL6814145 0.83 TRPA1 (0.52) MMP13TRPA1EPHX2PDE10AWDR5
SCHEMBL6819189 0.82 KDM5A (0.37) SCD
SCHEMBL6476888 0.77 RXRA (0.35)
SCHEMBL6814148 0.74 LOXL2 (0.40) MMP13TRPA1EPHX2
SCHEMBL6487515 0.74 MMP13 (0.46) MMP13TRPA1EPHX2CDK2GSK3B
SCHEMBL6822279 0.73 TRPA1 (0.47) MMP13TRPA1EPHX2PDE10AWDR5
SCHEMBL6814142 0.70 KDM5A (0.35) TRPA1SCD
SCHEMBL6477648 0.70 POLB (0.42) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014908-A1 HETEROBICYLCIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO claimed