SCHEMBL6814148

SCHEMBL6814148

COc1cc(CN)ccn1.Cc1c(=O)c(Cc2ccc(F)c(F)c2)cn2cc(C(=O)O)sc12

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 7/20 0.40
LOX P28300 4/20 0.40
TRPA1 O75762 1/20 0.38
GRM2 Q14416 1/20 0.34
EPHX2 P34913 1/20 0.32
KDM5A P29375 3/20 0.32
KDM5B Q9UGL1 3/20 0.32
KDM4C Q9H3R0 2/20 0.32
PLA2G7 Q13093 1/20 0.30
MMP13 P45452 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6814142 0.90 KDM5A (0.35) TRPA1GRM2KDM5AKDM5BKDM4C
SCHEMBL6814145 0.86 TRPA1 (0.52) TRPA1EPHX2MMP13
SCHEMBL6819195 0.85 LOXL2 (0.40) LOXL2LOXTRPA1GRM2KDM5A
SCHEMBL6484565 0.84 RXRA (0.35) TRPA1KDM5AKDM5B
SCHEMBL6819189 0.75 KDM5A (0.37) GRM2KDM5AKDM5BKDM4C
SCHEMBL6819192 0.74 MMP13 (0.41) TRPA1EPHX2MMP13
SCHEMBL6476858 0.72 TRPA1 (0.49) TRPA1
SCHEMBL6485426 0.70 P2RY14 (0.36) KDM5AKDM5B
Picolamine SCHEMBL6818607 0.68 PLA2G7 (0.34) TRPA1PLA2G7
SCHEMBL6476888 0.67 RXRA (0.35) KDM5AKDM5BKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014908-A1 HETEROBICYLCIC METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed