SCHEMBL6816973

SCHEMBL6816973

NC(=O)N(c1cccc(C(=O)O)c1)c1ccccc1Br

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA6 P23280 1/20 0.38
CA9 Q16790 1/20 0.38
AKR1C3 P42330 1/20 0.37
FABP4 P15090 1/20 0.37
FABP5 Q01469 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
DAO P14920 1/20 0.36
TSHR P16473 1/20 0.36
NAPRT Q6XQN6 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PARP1 P09874 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27576496 0.83 KMO (0.47) KMOCA12CA1CA2CA6
Biphenyl SCHEMBL27587719 0.81 HSD17B1 (0.36) AKR1C3ALDH1A1TSHRCYP2C9PARP1
SCHEMBL6820924 0.80 AKR1B1 (0.41) LMNATSHRCYP1A2HPGDPRSS1
SCHEMBL6812678 0.79 MRGPRX4 (0.42) KMOCA12CA1CA2CA6
SCHEMBL27558267 0.78 EGFR (0.37) CA12CA1CA2CA6CA9
SCHEMBL6920197 0.77 ALDH1A1 (0.41) CA12CA1CA2CA6CA9
SCHEMBL27587710 0.77 HSD17B1 (0.41) AKR1C3CYP2C9
SCHEMBL5210586 0.76 HTR1F (0.43)
SCHEMBL5612906 0.76 TTR (0.40) CA12CA1CA2CA6CA9
SCHEMBL7741614 0.74 NR4A2 (0.40) CA12CA1CA2CA6CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1185271-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2004-02-04 EP disclosed
CN-1356902-A IL-8 receptor antagonists SMITHKLINE BEECHAM CORP (US) 2002-07-03 CN disclosed
EP-1185271-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2002-03-13 EP disclosed
WO-2000076515-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2000-12-21 WO disclosed