SCHEMBL6920197

SCHEMBL6920197

NC(=O)N(c1ccc(Cl)c(C(=O)O)c1)c1ccccc1Br

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 3/20 0.39
KDM4E B2RXH2 3/20 0.39
POLB P06746 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 6/20 0.39
MEN1 O00255 5/20 0.39
LMNA P02545 1/20 0.38
GAA P10253 3/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA3 P07451 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6816973 0.77 KMO (0.39) ALDH1A1LMNACA12CA1CA2
SCHEMBL6820717 0.77 ALDH1A1 (0.51) ALDH1A1TP53MAPTKDM4EPOLB
SCHEMBL27576157 0.73 HNF4A (0.54) ALDH1A1MAPTKMT2ALMNAPTPN1
SCHEMBL27519456 0.72 MMP2 (0.44) ALDH1A1KDM4EKMT2ACA12CA1
Biphenyl SCHEMBL27587719 0.72 HSD17B1 (0.36) ALDH1A1NPC1RAB9APTPN1
SCHEMBL7611518 0.72 AKR1C3 (0.46) ALDH1A1KDM4EGLAPTPN1
SCHEMBL27587734 0.71 CXCR2 (0.45) KMT2AHPGDHSD17B10
SCHEMBL6820924 0.71 AKR1B1 (0.41) POLBLMNAGAAHPGDHTT
SCHEMBL27519344 0.71 CXCR2 (0.37) ALDH1A1TDP1
SCHEMBL5950300 0.70 ALDH1A1 (0.50) ALDH1A1TP53KDM4ERAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1185271-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2004-02-04 EP disclosed
CN-1356902-A IL-8 receptor antagonists SMITHKLINE BEECHAM CORP (US) 2002-07-03 CN disclosed
EP-1185271-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2002-03-13 EP disclosed
WO-2000076515-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2000-12-21 WO disclosed