SCHEMBL6833440

SCHEMBL6833440

COc1ccc2c(c1)c(CC(N)=O)cn2N=O

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 10/20 0.61
AKR1C3 P42330 5/20 0.50
AKR1C2 P52895 2/20 0.50
ICMT O60725 1/20 0.47
AKR1C4 P17516 1/20 0.46
PTGS1 P23219 1/20 0.46
PLA2G10 O15496 1/20 0.45
PTGS2 P35354 1/20 0.44
ADRB2 P07550 1/20 0.44
NQO2 P16083 1/20 0.44
MTNR1A P48039 1/20 0.44
MTNR1B P49286 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6833442 0.82 ADRB2 (0.67) ADRB2NQO2MTNR1AMTNR1B
SCHEMBL194360 0.78 MTNR1A (0.73) AKR1C3NQO2MTNR1AMTNR1B
SCHEMBL6938945 0.77 MTNR1A (0.58) AKR1C3NQO2MTNR1AMTNR1B
SCHEMBL6921381 0.77 MTNR1A (0.57) NQO2MTNR1AMTNR1B
SCHEMBL6921659 0.77 HTR6 (0.68) MTNR1A
SCHEMBL14041516 0.77 PLA2G2A (0.67) PLA2G2AICMT
SCHEMBL6944686 0.76 MTNR1A (0.57) NQO2MTNR1AMTNR1B
SCHEMBL6939654 0.76 MTNR1A (0.57) AKR1C3NQO2MTNR1AMTNR1B
SCHEMBL7963252 0.76 PLA2G2A (1.00) PLA2G2AICMTMTNR1AMTNR1B
SCHEMBL7122186 0.75 MTNR1A (0.55) AKR1C3NQO2MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004085392-A1 MELATONIN DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL DYSFUNCTIONS FAUST PHARMACEUTICALS (FR) 2004-10-07 WO disclosed
WO-2004085395-A1 MELATONIN DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL DYSFUNCTIONS FAUST PHARMACEUTICALS (FR) 2004-10-07 WO disclosed