SCHEMBL6833442

SCHEMBL6833442

COc1ccc2c(c1)c(CCN)cn2N=O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.67
HTR6 P50406 11/20 0.57
HTR2A P28223 2/20 0.47
CYP1A2 P05177 1/20 0.47
HTR1A P08908 1/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
NFKB1 P19838 1/20 0.47
HTR1D P28221 1/20 0.47
HTR1B P28222 1/20 0.47
HTR2C P28335 1/20 0.47
HTR7 P34969 1/20 0.47
HTR4 Q13639 1/20 0.47
TRPM8 Q7Z2W7 1/20 0.47
ADRA1A P35348 1/20 0.47
TAAR1 Q96RJ0 1/20 0.47
BLM P54132 1/20 0.46
PMP22 Q01453 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
MTNR1A P48039 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6921659 0.84 HTR6 (0.68) HTR6HTR1AHTR1DHTR1BHTR7
SCHEMBL6833440 0.82 PLA2G2A (0.61) ADRB2MTNR1ANQO2MTNR1B
SCHEMBL6949412 0.81 MTNR1A (0.49) ADRB2HTR6MTNR1ANQO2MTNR1B
SCHEMBL28121087 0.81 ADRB2 (0.67) ADRB2HTR6HTR2ACYP1A2HTR1A
SCHEMBL194360 0.80 MTNR1A (0.73) CYP1A2HTR1AHTR2CBLMPMP22
SCHEMBL1130016 0.80 ADRB2 (1.00) ADRB2HTR6HTR2ACYP1A2HTR1A
SCHEMBL6938945 0.79 MTNR1A (0.58) MTNR1ANQO2MTNR1B
SCHEMBL6919423 0.79 HTR6 (0.53) HTR6HTR1AHTR1DHTR1BHTR7
SCHEMBL6921381 0.79 MTNR1A (0.57) HTR6HTR1AHTR1DHTR1BHTR7
SCHEMBL10482825 0.79 ADRB2 (0.72) ADRB2HTR6HTR2ACYP1A2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004085392-A1 MELATONIN DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL DYSFUNCTIONS FAUST PHARMACEUTICALS (FR) 2004-10-07 WO disclosed
WO-2004085395-A1 MELATONIN DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL DYSFUNCTIONS FAUST PHARMACEUTICALS (FR) 2004-10-07 WO disclosed