Norfluoxetine

Norfluoxetine

SCHEMBL686500

NCCC(Oc1ccc(C(F)(F)F)cc1)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 1.00
SLC6A2 P23975 4/20 1.00
SLC6A3 Q01959 4/20 1.00
KCNK2 O95069 2/20 1.00
KCNH2 Q12809 2/20 1.00
CACNA1C Q13936 2/20 1.00
SLC7A5 Q01650 7/20 0.82
MEN1 O00255 4/20 0.68
KMT2A Q03164 4/20 0.68
LMNA P02545 4/20 0.68
HRH3 Q9Y5N1 2/20 0.68
NPC1 O15118 2/20 0.68
CYP2D6 P10635 2/20 0.68
CYP2C19 P33261 2/20 0.68
MTOR P42345 2/20 0.68
RAB9A P51151 2/20 0.68
CYP3A4 P08684 2/20 0.68
HTR2C P28335 2/20 0.68
KDM4E B2RXH2 1/20 0.68
TP53 P04637 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Seproxetine SCHEMBL272873 1.00 SLC6A4 (1.00) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
Norfluoxetine SCHEMBL3750512 1.00 SLC6A4 (1.00) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
Norfluoxetine SCHEMBL140929 0.98 SLC6A4 (0.97) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
Seproxetine SCHEMBL120303 0.98 SLC6A4 (0.97) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
Norfluoxetine SCHEMBL7306073 0.93 SLC6A4 (0.87) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
SCHEMBL17267513 0.90 SLC7A5 (1.00) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
SCHEMBL17267476 0.90 SLC7A5 (1.00) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
SCHEMBL17267474 0.90 SLC7A5 (1.00) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
SCHEMBL17267515 0.89 SLC7A5 (1.00) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
SCHEMBL2738930 0.88 SLC6A4 (0.78) SLC6A4SLC6A2SLC6A3KCNK2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 143 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3787631-B1 MODULATORS OF ORPHAN NUCLEAR RECEPTORS FOR NASH AND OTHER METABOLIC DISORDERS UNIV EMORY (US) 2025-09-10 EP claimed
EP-3603674-B1 COMBINATION OF MORPHINAN COMPOUNDS AND ANTIDEPRESSANT FOR THE TREATMENT OF INTRACTABLE AND CHRONIC PAIN SUN PHARMACEUTICAL IND INC (US) 2025-02-26 EP claimed
US-7485754-B2 Efficient method for preparing 3-aryloxy-3-arylpropylamines and their optical stereoisomers APOTEX PHARMACHEM INC. (CA) 2009-02-03 US claimed
WO-2007006132-A1 AN EFFICIENT METHOD FOR PREPARING 3-ARYLOXY-3- ARYLPROPYLAMINES AND THEIR OPTICAL STEREOISOMERS APOTEX PHARMACHEM INC. (CA) 2007-01-18 WO claimed
US-20070010678-A1 Efficient method for preparing 3-aryloxy-3-arylpropylamines and their optical stereoisomers APOTEX PHARMACHEM INC. 2007-01-11 US claimed
US-20040266882-A1 Aryloxypropylamines as chemosensitizing agents in the treatment of cancer RAMOT AT TEL AVIV UNIVERSITY LTD. (IL) 2004-12-30 US claimed
EP-1425002-A1 ARYLOXYPROPYLAMINES AS CHEMOSENSITIZING AGENTS IN THE TREATMENT OF CANCER Ramot at Tel Aviv University Ltd. (IL) 2004-06-09 EP claimed
US-20040054014-A1 Method and pharmaceutical compositions forthe treatment of cancer RAMOT AT TEL AVIV UNIVERSITY LTD. 2004-03-18 US claimed
US-6630454-B2 Method and pharmaceutical composition for the treatment of cancer RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2003-10-07 US claimed
US-20030087964-A1 Method and pharmaceutical composition for the treatment of cancer RAMOT UNIVERSITY AUTHORITY FOR APPLIED RESEARCH AND INDUSTRIAL DEVELOPMENT LTD. 2003-05-08 US claimed
EP-0831799-B1 COMPOUNDS ACTIVE AT A NOVEL SITE ON RECEPTOR-OPERATED CALCIUM CHANNELS USEFUL FOR TREATMENT OF NEUROLOGICAL DISORDERS NPS PHARMA INC (US) 2003-05-02 EP claimed
WO-2003022258-A1 ARYLOXYPROPYLAMINES AS CHEMOSENSITIZING AGENT IN THE TREATMENT OF CANCER RAMOT AT TEL AVIV UNIVERSITY LTD. (IL) 2003-03-20 WO claimed
EP-0969874-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING PROPANAMINE DERIVATIVES AND CYCLODEXTRIN Therabel Industries S.A. (FR) 2000-01-12 EP claimed
WO-1998042382-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING PROPANAMINE DERIVATIVES AND CYCLODEXTRIN THERABEL INDUSTRIES S.A. (FR) 1998-10-01 WO claimed
US-4313896-A ANTIDEPRESSANTS, PSYCHOTROPIC AGENTS ELI LILLY AND COMPANY (US) 1982-02-02 US claimed
US-4314081-A ANTIDEPRESSANTS ELI LILLY AND COMPANY (US) 1982-02-02 US claimed
CN-116283626-B Fluoxetine hapten, monoclonal antibody, hybridoma cell strain and application 江南大学 2024-12-06 CN disclosed
CN-118858475-A Detection reagent, detection kit and application thereof in psychotropic drug detection 广州凯普医学检验所有限公司 2024-10-29 CN disclosed
US-4194009-A ANTIDEPRESSANT ELI LILLY AND COMPANY (US) 1980-03-18 US disclosed
US-4018895-A Aryloxyphenylpropylamines in treating depression ELI LILLY AND COMPANY (US) 1977-04-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040054014-A1 Method and pharmaceutical compositions forthe treatment of cancer ABCC1, ABCB1, SLC11A2 SLC6A4 340/4885SLC6A2 374/4885SLC6A3 334/4885
US-20030087964-A1 Method and pharmaceutical composition for the treatment of cancer PNMT, ABCC1, HNMT SLC6A4 596/4885SLC6A2 550/4885SLC6A3 606/4885
US-20040266882-A1 Aryloxypropylamines as chemosensitizing agents in the treatment of cancer ABCC1, PNMT, ABCB1 SLC6A4 280/4885SLC6A2 290/4885SLC6A3 272/4885
US-20070010678-A1 Efficient method for preparing 3-aryloxy-3-arylpropylamines and their optical stereoisomers SLC6A4, HTR3A, TPH2 SLC6A4 1/4885SLC6A2 13/4885SLC6A3 12/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.