Norfluoxetine

Norfluoxetine

SCHEMBL3750512

NCC[C@@H](Oc1ccc(C(F)(F)F)cc1)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 1.00
SLC6A2 P23975 4/20 1.00
SLC6A3 Q01959 4/20 1.00
KCNK2 O95069 2/20 1.00
KCNH2 Q12809 2/20 1.00
CACNA1C Q13936 2/20 1.00
SLC7A5 Q01650 7/20 0.82
MEN1 O00255 4/20 0.68
KMT2A Q03164 4/20 0.68
LMNA P02545 4/20 0.68
HRH3 Q9Y5N1 2/20 0.68
NPC1 O15118 2/20 0.68
CYP2D6 P10635 2/20 0.68
CYP2C19 P33261 2/20 0.68
MTOR P42345 2/20 0.68
RAB9A P51151 2/20 0.68
CYP3A4 P08684 2/20 0.68
HTR2C P28335 2/20 0.68
KDM4E B2RXH2 1/20 0.68
TP53 P04637 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Seproxetine SCHEMBL272873 1.00 SLC6A4 (1.00) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
Norfluoxetine SCHEMBL686500 1.00 SLC6A4 (1.00) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
Norfluoxetine SCHEMBL140929 0.98 SLC6A4 (0.97) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
Seproxetine SCHEMBL120303 0.98 SLC6A4 (0.97) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
Norfluoxetine SCHEMBL7306073 0.93 SLC6A4 (0.87) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
SCHEMBL17267513 0.90 SLC7A5 (1.00) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
SCHEMBL17267476 0.90 SLC7A5 (1.00) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
SCHEMBL17267474 0.90 SLC7A5 (1.00) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
SCHEMBL17267515 0.89 SLC7A5 (1.00) SLC6A4SLC6A2SLC6A3KCNK2KCNH2
SCHEMBL2738930 0.88 SLC6A4 (0.78) SLC6A4SLC6A2SLC6A3KCNK2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7485754-B2 Efficient method for preparing 3-aryloxy-3-arylpropylamines and their optical stereoisomers APOTEX PHARMACHEM INC. (CA) 2009-02-03 US claimed
WO-2007006132-A1 AN EFFICIENT METHOD FOR PREPARING 3-ARYLOXY-3- ARYLPROPYLAMINES AND THEIR OPTICAL STEREOISOMERS APOTEX PHARMACHEM INC. (CA) 2007-01-18 WO claimed
US-20070010678-A1 Efficient method for preparing 3-aryloxy-3-arylpropylamines and their optical stereoisomers APOTEX PHARMACHEM INC. 2007-01-11 US claimed
CN-119120634-A Process for the preparation of (R) -oxiranes based on epoxide hydrolases 杭州微远生物科技有限公司 2024-12-13 CN disclosed
CN-118147265-B Chiral resolution method of oxirane compound based on epoxide hydrolase 杭州微远生物科技有限公司 2024-11-05 CN disclosed
CN-118147265-A Chiral resolution method of oxirane compound based on epoxide hydrolase 杭州微远生物科技有限公司 2024-06-07 CN disclosed
CN-111944774-B Alcohol dehydrogenase, encoding gene thereof and application of alcohol dehydrogenase in catalytic synthesis of (R) -styrene glycol 河北大学 2022-05-20 CN disclosed
US-20130123253-A1 MODULATORS OF CENTRAL NERVOUS SYSTEM NEUROTRANSMITTERS HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2013-05-16 US disclosed
US-8168635-B2 2-(aminomethyl)-5-phenyltetrahydrofuran; 4-(3,4-Dimethoxyphenyl)-2-[5-(2-{5-[2-(5-fluoro-2-methoxyphenyl)-ethyl]-tetrahydrofuran-2-yl}-ethylamino)-pentyl]-4a,5,8,8a-tetrahydro-2H-phthalazin-1-one; dual inhibitor of serotonin reuptake and phosphodiesterase 4 (PDE4) enzyme activity HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2012-05-01 US disclosed
US-20110136914-A1 SUBSTITUTED ARYLOXYPROPYLAMINES WITH SEROTONINERGIC AND/OR NOREPINEPHRINERGIC ACTIVITY AUSPEX PHARMACEUTICALS, INC. (US) 2011-06-09 US disclosed
US-20110136914-A1 SUBSTITUTED ARYLOXYPROPYLAMINES WITH SEROTONINERGIC AND/OR NOREPINEPHRINERGIC ACTIVITY AUSPEX PHARMACEUTICALS, INC. (US) 2011-06-09 US disclosed
US-20100292289-A1 TREATMENT OF METABOLIC SYNDROME WITH NOVEL AMIDES AMPLA PHARMACEUTICALS INC. (US) 2010-11-18 US disclosed
US-20100292289-A1 TREATMENT OF METABOLIC SYNDROME WITH NOVEL AMIDES AMPLA PHARMACEUTICALS INC. (US) 2010-11-18 US disclosed
US-20100292289-A1 TREATMENT OF METABOLIC SYNDROME WITH NOVEL AMIDES AMPLA PHARMACEUTICALS INC. (US) 2010-11-18 US disclosed
US-20080261967-A1 Modulators of Central Nervous System Neurotransmitters HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2008-10-23 US disclosed
US-20070155820-A1 SUBSTITUTED ARYLOXYPROPYLAMINES WITH SEROTONINERGIC AND/OR NOREPINEPHRINERGIC ACTIVITY AUSPEX PHARMACEUTICALS, INC. (US) 2007-07-05 US disclosed
US-20070155820-A1 SUBSTITUTED ARYLOXYPROPYLAMINES WITH SEROTONINERGIC AND/OR NOREPINEPHRINERGIC ACTIVITY AUSPEX PHARMACEUTICALS, INC. (US) 2007-07-05 US disclosed
WO-2007062119-A1 SUBSTITUTED ARYLOXYPROPYLAMINES WITH SEROTONINERGIC AND/OR NOREPINEPHRINERGIC ACTIVITY AUSPEX PHARMACEUTICALS, INC. (US) 2007-05-31 WO disclosed
US-20070078188-A1 Compositions comprising and methods of using norfluoxetine CURRIE MARK G 2007-04-05 US disclosed
US-20070078188-A1 Compositions comprising and methods of using norfluoxetine CURRIE MARK G 2007-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110136914-A1 SUBSTITUTED ARYLOXYPROPYLAMINES WITH SEROTONINERGIC AND/OR NOREPINEPHRINERGIC ACTIVITY SLC6A4, HTR4, GPR34 SLC6A4 1/4885SLC6A2 5/4885SLC6A3 17/4885
US-20080261967-A1 Modulators of Central Nervous System Neurotransmitters GAP43, SLC18A2, CHRNA6 SLC6A4 104/4885SLC6A2 47/4885SLC6A3 54/4885
US-20070155820-A1 SUBSTITUTED ARYLOXYPROPYLAMINES WITH SEROTONINERGIC AND/OR NOREPINEPHRINERGIC ACTIVITY SLC6A4, HTR4, GPR34 SLC6A4 1/4885SLC6A2 5/4885SLC6A3 17/4885
US-20070010678-A1 Efficient method for preparing 3-aryloxy-3-arylpropylamines and their optical stereoisomers SLC6A4, HTR3A, TPH2 SLC6A4 1/4885SLC6A2 13/4885SLC6A3 12/4885
US-20130123253-A1 MODULATORS OF CENTRAL NERVOUS SYSTEM NEUROTRANSMITTERS GAP43, SLC18A2, CHRNA6 SLC6A4 104/4885SLC6A2 47/4885SLC6A3 54/4885
US-20100292289-A1 TREATMENT OF METABOLIC SYNDROME WITH NOVEL AMIDES GPR119, CPT1A, GLS2 SLC6A4 1007/4885SLC6A2 962/4885SLC6A3 2178/4885
US-20070078188-A1 Compositions comprising and methods of using norfluoxetine ALOX5, NGF, PTGER4 SLC6A4 36/4885SLC6A2 70/4885SLC6A3 292/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.