SCHEMBL6870751

SCHEMBL6870751

Nc1cc(C(=O)NC2CCC2)cc2nc(-c3ccc[nH]3)nn12

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 11/20 0.41
HTT P42858 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MAP4K4 O95819 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
APOBEC3G Q9HC16 1/20 0.39
ABL1 P00519 1/20 0.39
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.37
KDR P35968 1/20 0.36
SMYD3 Q9H7B4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6868095 0.81 KDM4E (0.53) ADORA2AHTTKDM4EALDH1A1LMNA
SCHEMBL6870753 0.80 ADORA2A (0.37) ADORA2A
SCHEMBL6867019 0.80 DYRK1A (0.47) ADORA2AHTTKDM4EMAP4K4ALDH1A1
SCHEMBL6867472 0.79 ADORA2A (0.40) ADORA2A
SCHEMBL6863748 0.78 ADORA2A (0.64) ADORA2AHTTKDM4EALDH1A1LMNA
SCHEMBL6868478 0.78 ADORA2A (0.64) ADORA2AHTTKDM4EALDH1A1LMNA
SCHEMBL6868261 0.77 NPC1 (0.48) ADORA2AHTTKDM4EALDH1A1LMNA
SCHEMBL6870443 0.76 LMNA (0.45) ADORA2AKDM4EALDH1A1ABL1LMNA
SCHEMBL6869838 0.76 ADORA2A (0.43) ADORA2AHTTKDM4EALDH1A1LMNA
SCHEMBL6869677 0.75 ADORA2A (0.42) ADORA2AABL1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed