SCHEMBL6867944

SCHEMBL6867944

CN(C)c1ccnc(N[C@H]2CC[C@@H](NCc3cccc4ccccc34)CC2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.42
MCHR1 Q99705 1/20 0.42
ACHE P22303 7/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
TACR1 P25103 1/20 0.39
JAK3 P52333 1/20 0.38
BACE1 P56817 1/20 0.38
FLT3 P36888 1/20 0.38
TYRO3 Q06418 1/20 0.38
MERTK Q12866 1/20 0.38
GAS6 Q14393 1/20 0.38
MAPK8 P45983 3/20 0.37
MAPK9 P45984 3/20 0.37
MAPK10 P53779 3/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867978 1.00 ADRA2A (0.42) ADRA2AMCHR1ACHEMEN1KMT2A
SCHEMBL6869175 0.85 KDM1A (0.44) ADRA2AMCHR1ACHEJAK3BACE1
SCHEMBL6456622 0.85 SIGMAR1 (0.48) ADRA2AMCHR1ACHEALDH1A1
SCHEMBL6456613 0.85 SIGMAR1 (0.48) ADRA2AMCHR1ACHEALDH1A1
SCHEMBL6869183 0.85 KDM1A (0.44) ADRA2AMCHR1ACHEJAK3BACE1
SCHEMBL6867769 0.85 MEN1 (0.41) ADRA2AMCHR1ACHEMEN1KMT2A
SCHEMBL6867777 0.85 MEN1 (0.41) ADRA2AMCHR1ACHEMEN1KMT2A
SCHEMBL6875264 0.83 LMNA (0.54) ADRA2AMCHR1KMT2AMAPK8MAPK9
SCHEMBL6878043 0.83 SLC2A1 (0.43) ADRA2AMCHR1ACHEMEN1KMT2A
SCHEMBL6875616 0.82 KDM1A (0.46) ADRA2AMCHR1ACHEKMT2ABACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed