SCHEMBL6940743

SCHEMBL6940743

O=C(O)C(=O)CC(=O)c1cc(Cc2ccccc2)cc(N2CCN(Cc3ccccc3)CC2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.48
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
HTR2B P41595 1/20 0.47
DRD2 P14416 1/20 0.46
DRD3 P35462 1/20 0.46
ALDH1A1 P00352 3/20 0.46
HDAC4 P56524 2/20 0.45
HDAC1 Q13547 2/20 0.45
HDAC3 O15379 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HDAC9 Q9UKV0 1/20 0.45
HDAC5 Q9UQL6 1/20 0.45
HTR7 P34969 1/20 0.45
ITGB3 P05106 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6946070 0.87 PLOD2 (0.46) HTR2AHTR2CHTR2BMAPTMAPK1
SCHEMBL6950010 0.81 ALDH1A1 (0.50) ALDH1A1HDAC1KDM4EMAPTHTT
SCHEMBL6947604 0.78 ERCC5 (0.61) LMNA
SCHEMBL3348190 0.73 ALDH1A1 (0.58) DRD4HTR2AHTR2CHTR2BALDH1A1
SCHEMBL6949748 0.72 ERCC5 (0.53) ALDH1A1KDM4EHTTMEN1LMNA
SCHEMBL6940911 0.72 PTPN1 (0.72) KDM4EMAPTMEN1MAPK1KMT2A
SCHEMBL7671810 0.71 CYP19A1 (0.46)
SCHEMBL4021071 0.71 DRD2 (0.68) DRD4HTR2AHTR2CHTR2BDRD2
SCHEMBL6951304 0.71 ALDH1A1 (0.48) ALDH1A1HTTTSHRSMN1; SMN2
SCHEMBL6943565 0.71 L3MBTL1 (0.54) HTTLMNASMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed