SCHEMBL6946070

SCHEMBL6946070

CN1CCN(c2cc(Cc3ccccc3)cc(C(=O)CC(=O)C(=O)O)c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLOD2 O00469 1/20 0.46
PLOD3 O60568 1/20 0.46
PLOD1 Q02809 1/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
PTPN1 P18031 2/20 0.43
SIRT6 Q8N6T7 2/20 0.43
HTR6 P50406 4/20 0.43
ERCC5 P28715 1/20 0.42
FEN1 P39748 1/20 0.42
USP2 O75604 1/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
KMT2A Q03164 1/20 0.41
ESR2 Q92731 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6940743 0.87 DRD4 (0.48) MAPTMAPK1KMT2AHTR2AHTR2C
SCHEMBL7077276 0.84 LMNA (0.49) PLOD2PLOD3PLOD1NPC1RAB9A
SCHEMBL7078896 0.80 PLOD2 (0.47) PLOD2PLOD3PLOD1NPC1RAB9A
SCHEMBL6947604 0.79 ERCC5 (0.61) PTPN1ERCC5FEN1HAO1
SCHEMBL7667601 0.78 PIM2 (0.56) HRH2HRH1HRH3HRH4
SCHEMBL6949748 0.76 ERCC5 (0.53) NPC1RAB9APTPN1ERCC5FEN1
SCHEMBL7494302 0.74 ALDH1A1 (0.45) NPC1RAB9ASIRT6HTR6HTR1A
SCHEMBL7077564 0.73 AGXT (0.47) NPC1RAB9AHTR6ADRA2CHTR2A
Dimethylamine SCHEMBL6946035 0.73 PTPN1 (0.68) PTPN1ERCC5FEN1HAO1
SCHEMBL6946034 0.73 PTPN1 (0.53) PTPN1ERCC5FEN1KMT2ATMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed