SCHEMBL6969339

SCHEMBL6969339

CC(C)c1nc(CCOCc2ccccc2)n(Cc2ccc([N+](=O)[O-])cc2)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
PKM P14618 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
AR P10275 4/20 0.36
SLC29A1 Q99808 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
TDP1 Q9NUW8 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C9 P11712 2/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973218 0.94 CCR2 (0.41) ALDH1A1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL6962626 0.89 AGTR1 (0.34) ALDH1A1TDP1
SCHEMBL7084679 0.86 TDP1 (0.36) ALDH1A1TDP1CYP1A2CYP2C9CYP2D6
SCHEMBL6969108 0.84 TSHR (0.38) SMN1; SMN2ARMEN1KMT2ACYP1A2
SCHEMBL6962314 0.84 L3MBTL1 (0.36) ALDH1A1HPGDSMN1; SMN2ARMEN1
SCHEMBL14439828 0.84 TDP1 (0.40) SMN1; SMN2KMT2ATDP1NPC1RAB9A
SCHEMBL6961345 0.82 L3MBTL1 (0.39) ALDH1A1SMN1; SMN2ARMEN1KMT2A
SCHEMBL8349607 0.82 TDP1 (0.32) KMT2ATDP1
SCHEMBL6974526 0.82 TDP1 (0.32) ALDH1A1TDP1
SCHEMBL6972963 0.81 GSK3B (0.38) TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP claimed
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed