SCHEMBL6980758

SCHEMBL6980758

CCOC(=O)CCC(=O)N(Cc1ccccc1)c1cccc2c1N(C(=O)CCc1ccc(C#N)cc1)CCC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A1 P00352 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
MAPT P10636 2/20 0.36
NPC1 O15118 1/20 0.36
MAPK1 P28482 1/20 0.36
RAB9A P51151 1/20 0.36
USP14 P54578 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
LMNA P02545 2/20 0.35
GAA P10253 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
LTB4R2 Q9NPC1 1/20 0.35
TSHR P16473 2/20 0.35
AVPR2 P30518 1/20 0.35
OXTR P30559 1/20 0.35
AVPR1A P37288 1/20 0.35
CHRM2 P08172 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981595 0.90 LTB4R2 (0.46) ALDH1A1SMN1; SMN2MAPTNPC1MAPK1
SCHEMBL6982692 0.88 L3MBTL1 (0.38) NOTUML3MBTL1ALDH1A1SMN1; SMN2MAPT
SCHEMBL6986008 0.88 MEN1 (0.39) ALDH1A1SMN1; SMN2MAPTNPC1MAPK1
SCHEMBL6985399 0.86 NOTUM (0.36) NOTUML3MBTL1ALDH1A1SMN1; SMN2MAPT
SCHEMBL6980751 0.85 NOTUM (0.44) NOTUML3MBTL1ALDH1A1SMN1; SMN2MAPT
SCHEMBL6986002 0.84 RXRA (0.45) ALDH1A1SMN1; SMN2MAPTNPC1MAPK1
SCHEMBL6987767 0.82 TP53 (0.42) L3MBTL1ALDH1A1LMNAGAAUSP2
SCHEMBL6985613 0.82 CCR5 (0.37) NOTUML3MBTL1ALDH1A1SMN1; SMN2MAPT
SCHEMBL6987632 0.81 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2MAPTNPC1MAPK1
SCHEMBL6978045 0.81 ALDH1A1 (0.35) NOTUML3MBTL1ALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed