SCHEMBL6984759

SCHEMBL6984759

N#Cc1ccc(CCC(=O)N2CCCc3cccc(NS(=O)(=O)c4ccc(Cl)cc4)c32)cc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.47
ALDH1A1 P00352 4/20 0.47
GAA P10253 4/20 0.47
KDM4E B2RXH2 2/20 0.47
HTT P42858 1/20 0.47
TP53 P04637 3/20 0.40
PKM P14618 1/20 0.39
CCR2 P41597 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
NR3C1 P04150 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
GLO1 Q04760 1/20 0.37
MAPT P10636 1/20 0.37
THRB P10828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985322 0.92 GAA (0.41) LMNAALDH1A1GAATP53PKM
SCHEMBL6984039 0.92 TP53 (0.45) LMNAALDH1A1GAAKDM4EHTT
SCHEMBL7408050 0.92 TP53 (0.40) LMNAALDH1A1GAAKDM4EHTT
SCHEMBL6982764 0.92 FPR1 (0.43) LMNAALDH1A1GAAKDM4EPKM
SCHEMBL6985749 0.92 ALDH1A1 (0.48) LMNAALDH1A1GAAHTTTP53
SCHEMBL6981583 0.89 STAT3 (0.49) LMNAALDH1A1GAAHTTTP53
SCHEMBL6978217 0.89 SLC16A3 (0.42) LMNAALDH1A1HTTTP53PKM
SCHEMBL6982953 0.89 CCR10 (0.39) LMNAALDH1A1GAATP53PKM
SCHEMBL6982163 0.88 SLC16A3 (0.45) LMNAALDH1A1GAAHTTTP53
SCHEMBL6977498 0.87 CCKBR (0.44) LMNAALDH1A1GAATP53PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed