SCHEMBL6983872

SCHEMBL6983872

CCCN(CCCCN1CCCCC1=O)CC(C)c1cccc(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MC4R P32245 1/20 0.42
HTR7 P34969 2/20 0.39
DRD3 P35462 1/20 0.38
KCNH2 Q12809 1/20 0.38
ADRA1B P35368 1/20 0.37
UBE2M P61081 3/20 0.37
DCUN1D1 Q96GG9 3/20 0.37
ELANE P08246 2/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
KCNQ2 O43526 1/20 0.35
KMT2A Q03164 1/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSK P43235 1/20 0.35
PDK2 Q15119 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6977704 0.89 HTR7 (0.40) MC4RHTR7DRD3KCNH2ADRA1B
SCHEMBL6982527 0.88 NPC1 (0.41) ADRA1BGAARAB9AKMT2A
SCHEMBL4875623 0.79 HTR2A (0.39) HTR7DRD3UBE2MDCUN1D1ELANE
SCHEMBL6985684 0.77 ADRA1B (0.47) MC4RADRA1B
SCHEMBL4870508 0.77 HTR2A (0.40) HTR7DRD3ELANEGAAKMT2A
SCHEMBL6983282 0.77 LMNA (0.45) ADRA1BRAB9AKMT2A
SCHEMBL6987894 0.77 ADRA1B (0.37) ADRA1BKMT2A
SCHEMBL6983790 0.76 KMT2A (0.39) ADRA1BKMT2A
SCHEMBL6983291 0.76 ADRA1B (0.32) ADRA1B
SCHEMBL6979847 0.76 ADRA1B (0.41) ADRA1BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289965-A1 SUBSTITUTED 1-AMINOALKYL-LACTAMS AND THEIR USE AS MUSCARINIC RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2003-03-12 EP disclosed
WO-2001090081-A1 SUBSTITUTED 1-AMINOALKYL-LACTAMS AND THEIR USE AS MUSCARINIC RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-11-29 WO disclosed