SCHEMBL6986054

SCHEMBL6986054

COc1cc(N(C)C(=O)CCCN2CCN3CCCCC3C2)cc(OC)c1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.46
SHMT2 P34897 2/20 0.43
SLC29A1 Q99808 5/20 0.40
LMNA P02545 3/20 0.40
CYP2D6 P10635 2/20 0.40
KCNH2 Q12809 2/20 0.40
HRH3 Q9Y5N1 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ATM Q13315 1/20 0.40
POLB P06746 1/20 0.40
ABCC4 O15439 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
CHRM3 P20309 1/20 0.40
HTR2A P28223 1/20 0.40
MAPK1 P28482 1/20 0.40
SLC6A4 P31645 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5842883 0.99 SIGMAR1 (0.46) SIGMAR1SHMT2SLC29A1LMNACYP2D6
SCHEMBL6986839 0.86 ALDH1A1 (0.43) SIGMAR1SHMT2SLC29A1LMNAATM
SCHEMBL5842277 0.84 SLC29A1 (0.42) SIGMAR1SLC29A1MEN1KMT2A
SCHEMBL6984251 0.82 HTR7 (0.41) SIGMAR1SHMT2KCNH2CHRM3ADRA2A
SCHEMBL6986270 0.82 SLC29A1 (0.41) SIGMAR1SHMT2SLC29A1LMNACYP2D6
SCHEMBL6986043 0.82 SHMT2 (0.50) SHMT2SLC29A1LMNASMN1; SMN2ATM
Hydrochloric Acid SCHEMBL5840216 0.81 HTR7 (0.41) SIGMAR1KCNH2CHRM3ADRA2AADRA2C
Hydrochloric Acid SCHEMBL5842572 0.81 MEN1 (0.40) SIGMAR1SHMT2SLC29A1LMNACYP2D6
Hydrochloric Acid SCHEMBL5843596 0.81 SHMT2 (0.49) SHMT2LMNASMN1; SMN2ATMPOLB
SCHEMBL6984898 0.78 SLC29A1 (0.69) SLC29A1KCNH2MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1275647-B1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-11-12 EP disclosed
EP-1275647-A1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2003-01-15 EP disclosed