SCHEMBL6986371

SCHEMBL6986371

CC(C)n1nc(-c2cc(O)nn2-c2ccccc2)ccc1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.36
BMPR1B O00238 1/20 0.36
BMPR1A P36894 1/20 0.36
TGFBR1 P36897 1/20 0.36
ACVRL1 P37023 1/20 0.36
ACVR1 Q04771 1/20 0.36
MDM2 Q00987 2/20 0.36
MCL1 Q07820 2/20 0.36
TSHR P16473 1/20 0.36
BCL2 P10415 1/20 0.36
TP53 P04637 1/20 0.36
RPA1 P27694 1/20 0.36
POLB P06746 2/20 0.36
HSD11B1 P28845 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
MAPK1 P28482 1/20 0.35
GRN P28799 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6987355 0.85 ALDH1A1 (0.38) ALDH1A1GAAKMT2ABMPR1BBMPR1A
SCHEMBL6986812 0.82 ALDH1A1 (0.40) ALDH1A1GAAKMT2AMDM2MCL1
SCHEMBL6985846 0.81 BCL2 (0.41) ALDH1A1GAAKMT2AMDM2MCL1
SCHEMBL6985626 0.81 SLC5A1 (0.43) TSHRTP53NPC1RAB9AHTT
SCHEMBL6982469 0.81 CYP2C9 (0.39) ALDH1A1GAAKMT2AMDM2MCL1
SCHEMBL6985081 0.80 SLC5A1 (0.42) ALDH1A1TP53POLBNPC1RAB9A
SCHEMBL6981026 0.80 AGTR2 (0.40) ALDH1A1KMT2ATSHRTP53HSD11B1
SCHEMBL6984657 0.80 GRM5 (0.35) ALDH1A1GAABMPR1BBMPR1ATGFBR1
SCHEMBL6987183 0.80 TSHR (0.45) ALDH1A1MDM2MCL1TSHRBCL2
SCHEMBL6983748 0.79 GRM5 (0.46) ALDH1A1GAAKMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313733-A1 PYRAZOLOPYRIDINE COMPOUND AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-05-28 EP disclosed
WO-2002018382-A1 PYRAZOLOPYRIDINE COMPOUND AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-03-07 WO disclosed