SCHEMBL6986817

SCHEMBL6986817

N#Cc1ccc(CCC(=O)N2CCCc3cccc(NC(=O)Cc4ccccc4)c32)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.42
ATM Q13315 1/20 0.42
LMNA P02545 2/20 0.41
KMT2A Q03164 2/20 0.41
KCNQ2 O43526 1/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
RORC P51449 1/20 0.40
TP53 P04637 1/20 0.40
FPR1 P21462 2/20 0.40
FPR2 P25090 2/20 0.40
POLB P06746 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985381 0.88 MMP1 (0.45) ATMKMT2AFPR1FPR2POLB
SCHEMBL6980994 0.87 RXRA (0.43) ATMKMT2ATP53FPR1FPR2
SCHEMBL6986437 0.85 PTGER4 (0.41) ATMKMT2ATP53FPR1FPR2
SCHEMBL6985566 0.85 PARP14 (0.40) ATMKMT2ATP53FPR1FPR2
SCHEMBL6984462 0.84 ATM (0.41) ATMKMT2AGAARORCFPR1
SCHEMBL6977736 0.83 CHRM3 (0.40) ATMKMT2AFPR1FPR2ALDH1A1
SCHEMBL6985322 0.83 GAA (0.41) THRBLMNAKMT2AGAAPKM
SCHEMBL6983660 0.83 PTGER4 (0.40) KMT2AFPR1FPR2ALDH1A1MAPT
SCHEMBL6986809 0.82 RAB9A (0.51) THRBLMNARORCTP53FPR1
SCHEMBL7407513 0.81 RAB9A (0.44) KMT2AGAAFPR1FPR2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed