SCHEMBL6997801

SCHEMBL6997801

Cn1ccc2c1C(=O)N(CCCCBr)CCC2=O

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 7/20 0.32
DRD2 P14416 7/20 0.32
DRD1 P21728 4/20 0.32
DRD4 P21917 1/20 0.32
GRM5 P41594 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HTR1A P08908 3/20 0.31
HTR2A P28223 3/20 0.31
PNMT P11086 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7144008 0.85 DRD3 (0.33) DRD3DRD2DRD1DRD4GRM5
SCHEMBL6996046 0.85 KDM4E (0.33) DRD3DRD2DRD1DRD4GRM5
SCHEMBL6992176 0.79 TBXAS1 (0.43)
SCHEMBL6990341 0.78 DRD3 (0.54) DRD3DRD2DRD1DRD4HTR1A
SCHEMBL6989349 0.77 SIGMAR1 (0.47) DRD3DRD2DRD4TSHRHTR1A
SCHEMBL6994421 0.76 HTR1A (0.53) DRD3DRD2DRD1DRD4HTR1A
SCHEMBL6994882 0.76 PTPN1 (0.31) PNMT
SCHEMBL6774144 0.76 DRD3 (0.36) DRD3DRD2DRD1DRD4GRM5
SCHEMBL6989751 0.75 PNMT (0.32) PNMT
SCHEMBL6988025 0.74 L3MBTL1 (0.39) GRM5SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0557526-B1 PYRROLOAZEPINE COMPOUND SUNTORY LTD (JP) 2003-04-02 EP disclosed
US-5399557-A Cardiovascular disorders SUNTORY LIMITED (JP) 1995-03-21 US disclosed
EP-0557526-A1 PYRROLOAZEPINE COMPOUND SUNTORY LIMITED (JP) 1993-09-01 EP disclosed