SCHEMBL7017597

SCHEMBL7017597

O=c1c2ccccc2nc(C(Cl)Cl)n1-c1ccc(C(O)(C(F)(F)F)C(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 9/20 0.44
TP53 P04637 1/20 0.43
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GFER P55789 1/20 0.41
MLYCD O95822 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7020798 0.88 KCNH2 (0.50) CXCR3TP53MLYCD
SCHEMBL7016853 0.85 MLYCD (0.43) CXCR3TP53MAPK1ALDH1A1MLYCD
SCHEMBL7100648 0.83 CXCR3 (0.44) CXCR3ALDH1A1MLYCD
SCHEMBL7018385 0.82 TP53 (0.46) TP53MAPK1SMN1; SMN2ALDH1A1
SCHEMBL7016812 0.82 TP53 (0.46) TP53MAPK1SMN1; SMN2ALDH1A1
SCHEMBL7014520 0.81 ALDH1A1 (0.52) MAPK1SMN1; SMN2ALDH1A1
SCHEMBL7100250 0.81 MEN1 (0.60) TP53ALDH1A1
SCHEMBL7013568 0.80 LMNA (0.53) MAPK1SMN1; SMN2ALDH1A1
SCHEMBL7023261 0.78 ALDH1A1 (0.70) MAPK1SMN1; SMN2ALDH1A1
SCHEMBL7023859 0.77 ALDH1A1 (0.56) MAPK1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003106435-A1 FUSED-RING PYRIMIDIN-4(3H)-ONE DERIVATIVES, PROCESSES FOR THE PREPARATION AND USES THEREOF SANKYO COMPANY, LIMITED (JP) 2003-12-24 WO disclosed