SCHEMBL7020798

SCHEMBL7020798

CC(C)c1nc2ccccc2c(=O)n1-c1ccc(C(O)(C(F)(F)F)C(F)(F)F)cc1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.50
HRH3 Q9Y5N1 1/20 0.50
MLYCD O95822 7/20 0.49
CXCR3 P49682 7/20 0.48
TRPV1 Q8NER1 1/20 0.47
TP53 P04637 1/20 0.46
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7017597 0.88 CXCR3 (0.44) MLYCDCXCR3TP53
SCHEMBL7016853 0.85 MLYCD (0.43) MLYCDCXCR3TP53
SCHEMBL7100648 0.83 CXCR3 (0.44) MLYCDCXCR3
SCHEMBL6979418 0.82 KCNH2 (0.59) KCNH2HRH3TRPV1ESR1ESR2
SCHEMBL7016812 0.82 TP53 (0.46) TP53
SCHEMBL7018385 0.82 TP53 (0.46) TP53
SCHEMBL7100250 0.81 MEN1 (0.60) KCNH2HRH3TP53
SCHEMBL7021106 0.80 ALDH1A1 (0.57) CXCR3
SCHEMBL7104431 0.80 ALDH1A1 (0.50) TP53
SCHEMBL7014520 0.79 ALDH1A1 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003106435-A1 FUSED-RING PYRIMIDIN-4(3H)-ONE DERIVATIVES, PROCESSES FOR THE PREPARATION AND USES THEREOF SANKYO COMPANY, LIMITED (JP) 2003-12-24 WO disclosed