SCHEMBL7044003

SCHEMBL7044003

N#Cc1c(F)c(F)cc(C(N)=O)c1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.38
TRPV4 Q9HBA0 1/20 0.35
CES2 O00748 2/20 0.34
CES1 P23141 2/20 0.34
STAT3 P40763 2/20 0.34
PARP1 P09874 2/20 0.33
CYP11B2 P19099 1/20 0.33
ROCK2 O75116 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
CASP1 P29466 1/20 0.32
AURKA O14965 1/20 0.32
RPS6KB1 P23443 1/20 0.32
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA4 P22748 1/20 0.31
TAS1R3 Q7RTX0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5364750 0.85 TRPV4 (0.38) TRPV4CES2CES1STAT3KDM4E
SCHEMBL3552234 0.83 KEAP1 (0.39) TRPV4CES2CES1STAT3KDM4E
SCHEMBL5362826 0.83 ALDH1A1 (0.39) TRPV4CES2CES1STAT3KDM4E
SCHEMBL14408161 0.81 STAT3 (0.36) TRPV4CES2CES1STAT3CYP11B2
SCHEMBL7045129 0.79 ALDH1A1 (0.48) STAT3KDM4EALDH1A1HPGDCA1
SCHEMBL28085635 0.76 DGAT1 (0.45) DGAT1CES2CES1PARP1ROCK2
SCHEMBL829400 0.76 DGAT1 (0.45) DGAT1CES2CES1PARP1ROCK2
SCHEMBL7038698 0.75 CASP1 (0.39) DGAT1TRPV4PARP1CYP11B2ROCK2
SCHEMBL809118 0.75 TRPV4 (0.50) TRPV4CES2CES1STAT3CA1
SCHEMBL3552211 0.74 STAT3 (0.56) STAT3KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001929-B1 METHOD FOR PREPARING 3-CYANO-2,4-DIHALOGEN-5-FLUOR-BENZOIC ACID BAYER AG (DE) 2003-03-26 EP disclosed
US-6462218-B1 BY HYDROLYTIC CLEAVAGE CARRIED OUT IN THE PRESENCE OF ACIDS AND WATER OF ITS AMIDE, ESTER OR CYANO DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2002-10-08 US disclosed
EP-1001929-A1 METHOD FOR PREPARING 3-CYANO-2,4-DIHALOGEN-5-FLUOR-BENZOIC ACID Bayer Aktiengesellschaft (DE) 2000-05-24 EP disclosed
WO-1999006360-A1 METHOD FOR PREPARING 3-CYANO-2,4-DIHALOGEN-5-FLUOR-BENZOIC ACID BAYER AKTIENGESELLSCHAFT (DE) 1999-02-11 WO disclosed