SCHEMBL7062957

SCHEMBL7062957

CC(C)(C)ON(C=O)NCc1cc2ccccc2s1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.50
ADRB2 P07550 1/20 0.50
AGXT P21549 1/20 0.40
ASIC3 Q9UHC3 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.40
HDAC1 Q13547 1/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
PTGS2 P35354 2/20 0.36
S1PR4 O95977 3/20 0.36
S1PR5 Q9H228 3/20 0.36
IDH1 O75874 1/20 0.34
GLS O94925 1/20 0.34
FAAH O00519 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5373022 0.74 ADH1B (0.42) MEN1KMT2A
SCHEMBL1176902 0.70 CYP2A6 (0.62) CYP2A6ADRB2AGXTASIC3LOXL2
SCHEMBL15961524 0.70 CYP2A6 (0.67) CYP2A6ADRB2AGXTASIC3LOXL2
SCHEMBL7059655 0.69 TSHR (0.41) MEN1KMT2A
SCHEMBL27470182 0.69 CYP2A6 (0.56) CYP2A6ADRB2AGXTASIC3LOXL2
SCHEMBL7061210 0.69 SMN1; SMN2 (0.42) MEN1KMT2A
SCHEMBL1254283 0.68 CYP2A6 (1.00) CYP2A6ADRB2AGXTASIC3LOXL2
SCHEMBL5767231 0.68 CHRM2 (0.44) MEN1KMT2A
SCHEMBL7061205 0.66 RAB9A (0.40)
SCHEMBL6762362 0.66 RIPK1 (0.37) MEN1KMT2AKDM4CPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030162783-A1 Method and composition for the treatment of pain ASTRAZENECA AB (SE) 2003-08-28 US disclosed
EP-1248621-A1 METHOD AND COMPOSITION FOR THE TREATMENT OF PAIN AstraZeneca AB (SE) 2002-10-16 EP disclosed
WO-2001047523-A1 METHOD AND COMPOSITION FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2001-07-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030162783-A1 Method and composition for the treatment of pain OPRK1, OPRD1, ACHE CYP2A6 394/4885ADRB2 44/4885AGXT 2619/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.