SCHEMBL7083579

SCHEMBL7083579

CC(C)c1nc(COC(N)=O)n(Cc2ccccc2N)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
MAPK1 P28482 1/20 0.32
P2RX3 P56373 1/20 0.31
EPHX1 P07099 1/20 0.31
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6964951 0.91 ALDH1A1 (0.32) ALDH1A1POLBMAPK1P2RX3
SCHEMBL6957642 0.90 ALDH1A1 (0.34) ALDH1A1POLBMAPK1
SCHEMBL6973336 0.89 ALDH1A1 (0.32) ALDH1A1POLBMAPK1EPHX1
SCHEMBL6967638 0.89 TDP1 (0.39) ALDH1A1POLBP2RX3TDP1
SCHEMBL6965901 0.87 RAB9A (0.35) TDP1
SCHEMBL6972846 0.86 P2RX3 (0.34) ALDH1A1P2RX3TDP1
SCHEMBL6962617 0.86 P2RX3 (0.35) P2RX3
SCHEMBL6960543 0.86 GCGR (0.33) ALDH1A1TDP1
SCHEMBL14001658 0.85 P2RX3 (0.35) P2RX3TDP1
SCHEMBL6966022 0.85 ADRA1D (0.36) ALDH1A1MAPK1P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed