SCHEMBL6964951

SCHEMBL6964951

CC(C)c1nc(CCOC(N)=O)n(Cc2ccccc2N)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
POLB P06746 1/20 0.32
MAPK1 P28482 1/20 0.32
P2RX3 P56373 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6957642 0.95 ALDH1A1 (0.34) ALDH1A1KDM4ELMNAHPGDSMN1; SMN2
SCHEMBL7083579 0.91 ALDH1A1 (0.32) ALDH1A1POLBMAPK1P2RX3
SCHEMBL6960825 0.90 ALDH1A1 (0.32) ALDH1A1POLBMAPK1
SCHEMBL6960943 0.88 AGTR1 (0.35) ALDH1A1KDM4ELMNA
SCHEMBL7081352 0.87 TDP1 (0.31) SMN1; SMN2
SCHEMBL6966285 0.87 P2RX3 (0.33) ALDH1A1KDM4EHPGDSMN1; SMN2P2RX3
SCHEMBL6969846 0.86 KDM4E (0.33) ALDH1A1KDM4ELMNAHPGDSMN1; SMN2
SCHEMBL7084635 0.85 ADRA1D (0.35) ALDH1A1KDM4EHPGDSMN1; SMN2MAPK1
SCHEMBL6973223 0.85 TDP1 (0.33) ALDH1A1KDM4ELMNAHPGDSMN1; SMN2
SCHEMBL6973396 0.85 PIM1 (0.34) P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed