SCHEMBL7166019

SCHEMBL7166019

COc1cccc(C(=O)CCc2ccccc2)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.69
NPC1 O15118 2/20 0.69
MAPT P10636 2/20 0.65
TDP1 Q9NUW8 2/20 0.65
ALDH1A1 P00352 1/20 0.65
GPR52 Q9Y2T5 1/20 0.63
HSD11B1 P28845 2/20 0.59
GAA P10253 2/20 0.59
CES2 O00748 1/20 0.57
CES1 P23141 1/20 0.57
HTR1A P08908 1/20 0.56
ADRA2A P08913 1/20 0.56
DRD1 P21728 1/20 0.56
SLC6A2 P23975 1/20 0.56
SLC6A4 P31645 1/20 0.56
ADRA1A P35348 1/20 0.56
OPRM1 P35372 1/20 0.56
DRD3 P35462 1/20 0.56
SLC6A3 Q01959 1/20 0.56
KCNH2 Q12809 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9320692 0.93 RAB9A (0.64) RAB9ANPC1MAPTTDP1ALDH1A1
SCHEMBL27628173 0.91 RAB9A (0.69) RAB9ANPC1MAPTTDP1ALDH1A1
SCHEMBL8269548 0.89 HSD11B1 (0.64) RAB9ANPC1TDP1ALDH1A1HSD11B1
SCHEMBL7868068 0.87 RAB9A (0.56) RAB9ANPC1MAPTTDP1ALDH1A1
SCHEMBL1515775 0.86 MEN1 (0.61) RAB9ANPC1TDP1GPR52HSD11B1
SCHEMBL30416831 0.84 ALDH1A1 (0.69) RAB9ANPC1MAPTTDP1ALDH1A1
SCHEMBL4722288 0.84 ALDH1A1 (0.69) RAB9ANPC1MAPTTDP1ALDH1A1
SCHEMBL14306005 0.83 ALDH1A1 (0.60) RAB9ANPC1MAPTTDP1ALDH1A1
SCHEMBL7195774 0.82 MAPT (0.56) MAPTTDP1ALDH1A1HSD11B1CES2
SCHEMBL1304210 0.82 NPC1 (1.00) RAB9ANPC1MAPTALDH1A1GPR52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106478395-B A kind of method of iridium catalyzed synthesizing alpha-alkyl ketone 南京理工大学 2019-06-25 CN disclosed
CN-106478395-A A kind of method of iridium catalyzed synthesizing alpha-alkyl ketone 南京理工大学 2017-03-08 CN disclosed
CN-105906543-A Novel synthesis method of multifunctional pyrrole 常州大学 2016-08-31 CN disclosed
US-6653508-B2 Use treating various medical conditions, including pain GRUENENTHAL GMBH (DE) 2003-11-25 US disclosed
US-20020161262-A1 3-Amino-2-benzyl-1-phenylpropane derivatives GRUENTENTHAL GMBH (DE) 2002-10-31 US disclosed
EP-1196373-A1 3-AMINO-2-BENZYL-1-PHENYL-PROPANE DERIVATIVES Grünenthal GmbH (DE) 2002-04-17 EP disclosed
WO-2001005743-A1 3-AMINO-2-BENZYL-1-PHENYL-PROPANE DERIVATIVES Grünenthal GmbH (DE) 2001-01-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020161262-A1 3-Amino-2-benzyl-1-phenylpropane derivatives PYGL, CYP11B2, GOT2 RAB9A 1573/4885NPC1 11/4885MAPT 1038/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.