SCHEMBL7200638

SCHEMBL7200638

CCN(CCCCN1CCN(S(=O)(=O)C(N)CCc2ccccc2)CC1=O)C(C)Cc1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.34
SIGMAR1 Q99720 1/20 0.34
ACHE P22303 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MCL1 Q07820 1/20 0.34
RORC P51449 2/20 0.33
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
PKM P14618 1/20 0.32
CCR5 P51681 8/20 0.32
KCNH2 Q12809 2/20 0.32
CHRM5 P08912 1/20 0.31
CHRM1 P11229 1/20 0.31
DPP4 P27487 1/20 0.31
CCR2 P41597 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7158802 0.88 LMNA (0.30)
SCHEMBL7200643 0.86 PKM (0.33) SIGMAR1ACHERORCALDH1A1GAA
SCHEMBL7085854 0.85 CCR2 (0.33) TSHRSIGMAR1ACHEKDM4EMCL1
SCHEMBL4875121 0.84 CYP2D6 (0.36) TSHRRORCSLC6A2SLC6A4SLC6A3
SCHEMBL4874460 0.84 ACHE (0.33) TSHRSIGMAR1ACHEKDM4EMCL1
SCHEMBL27492225 0.83 TSHR (0.33) TSHRSIGMAR1KDM4EMCL1RORC
SCHEMBL7158804 0.82 CCR5 (0.30) CCR5
SCHEMBL4874473 0.81 MAOB (0.34) SIGMAR1ACHERORCALDH1A1GAA
SCHEMBL4871446 0.81 CCR5 (0.35) SIGMAR1ACHERORCALDH1A1GAA
SCHEMBL4873613 0.81 LMNA (0.31) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289965-A1 SUBSTITUTED 1-AMINOALKYL-LACTAMS AND THEIR USE AS MUSCARINIC RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2003-03-12 EP disclosed
WO-2001090081-A1 SUBSTITUTED 1-AMINOALKYL-LACTAMS AND THEIR USE AS MUSCARINIC RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-11-29 WO disclosed