SCHEMBL7201786

SCHEMBL7201786

COc1ccccc1C1CCN(S(=O)(=O)C2CCNCC2(O)C(=O)NO)CC1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 3/20 0.49
MMP13 P45452 2/20 0.49
MMP9 P14780 1/20 0.49
HTR2C P28335 2/20 0.46
MEN1 O00255 5/20 0.44
KMT2A Q03164 5/20 0.44
ADAM10 O14672 1/20 0.42
MAPT P10636 1/20 0.42
CHRM4 P08173 2/20 0.40
CHRM1 P11229 2/20 0.40
CHRM2 P08172 1/20 0.40
MCOLN2 Q8IZK6 1/20 0.40
MCOLN3 Q8TDD5 1/20 0.40
MCOLN1 Q9GZU1 1/20 0.40
DRD2 P14416 2/20 0.39
DRD4 P21917 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7205516 0.87 ADAM10 (0.51) MMP2MMP13HTR2CADAM10DRD4
SCHEMBL7202570 0.86 EPHX2 (0.41) MMP2MMP13MMP9HTR2CMEN1
SCHEMBL7201770 0.85 MMP2 (0.44) MMP2MMP13MMP9ADAM10CHRM4
SCHEMBL7204290 0.85 MMP2 (0.46) MMP2MMP13ADAM10
SCHEMBL7205207 0.84 MMP13 (0.54) MMP2MMP13MMP9MEN1KMT2A
SCHEMBL7201610 0.83 MMP2 (0.47) MMP2MMP13MMP9ADAM10
SCHEMBL7208003 0.83 ALDH1A1 (0.41) MMP2MMP13MEN1KMT2AMAPT
SCHEMBL7207178 0.82 USP5 (0.43) MMP2MMP13MMP9
SCHEMBL7204170 0.81 HTR2C (0.48) MMP2MMP13MMP9HTR2CADAM10
SCHEMBL7201577 0.81 MMP1 (0.42) MMP2MMP13HTR2CMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6608104-B2 Antiarthritic agents; anticancer agents PFIZER INC 2003-08-19 US disclosed
US-20020019534-A1 Gem substituted hydroxamic acids PFIZER INC. 2002-02-14 US disclosed
EP-1138680-A1 Gem substituted sulfonyl hydroxamic acids as MMP inhibitors Pfizer Products Inc. (US) 2001-10-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020019534-A1 Gem substituted hydroxamic acids MMP14, TOP2A, ADAMTS1 MMP2 13/4885MMP13 4/4885MMP9 24/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.