SCHEMBL7207784

SCHEMBL7207784

COc1ccc(S(=O)(=O)C(c2ccccc2)C(C)C(=O)O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 8/20 0.54
MMP3 P08254 7/20 0.54
PDE4A P27815 6/20 0.54
PDE4B Q07343 6/20 0.54
PDE4C Q08493 6/20 0.54
PDE4D Q08499 6/20 0.54
MMP1 P03956 7/20 0.54
MMP13 P45452 5/20 0.52
MMP9 P14780 5/20 0.51
MMP8 P22894 2/20 0.51
MMP12 P39900 1/20 0.51
MMP14 P50281 1/20 0.51
MMP16 P51512 1/20 0.51
NPC1 O15118 2/20 0.49
ALDH1A1 P00352 2/20 0.49
RAB9A P51151 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
TDP1 Q9NUW8 1/20 0.49
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7515598 0.87 SMN1; SMN2 (0.51) MMP2MMP3PDE4APDE4BPDE4C
SCHEMBL7207035 0.80 MMP1 (0.54) MMP2MMP3PDE4APDE4BPDE4C
SCHEMBL15617672 0.79 NPC1 (0.58) MMP2MMP3PDE4APDE4BPDE4C
SCHEMBL7352846 0.77 MMP13 (0.60) MMP2MMP3PDE4APDE4BPDE4C
SCHEMBL8713229 0.75 MMP1 (0.58) MMP2MMP3PDE4APDE4BPDE4C
SCHEMBL6929276 0.74 MMP1 (0.70) MMP2MMP3PDE4APDE4BPDE4C
SCHEMBL8014627 0.74 MMP2 (0.78) MMP2MMP3PDE4APDE4BPDE4C
SCHEMBL28548434 0.74 NPC1 (0.54) MMP2MMP3PDE4APDE4BPDE4C
SCHEMBL7212138 0.73 MMP13 (0.54) MMP2MMP3PDE4APDE4BPDE4C
SCHEMBL7207763 0.72 MMP1 (0.49) MMP2MMP3PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0939628-B1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 2003-03-05 EP disclosed
US-6013649-A BOND DISORDERS; AUTOIMMUNE DISEASES; ANTITUMOR AGENTS MONSANTO COMPANY (US) 2000-01-11 US disclosed
EP-0939628-A4 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 1999-12-22 EP disclosed
EP-0939628-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1999-09-08 EP disclosed
WO-1998003164-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1998-01-29 WO disclosed