SCHEMBL7239090

SCHEMBL7239090

CCOC(=O)CC(c1ccccc1)n1ccc2cc[nH]c2c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
KDM4E B2RXH2 3/20 0.40
HTT P42858 2/20 0.40
BRD4 O60885 1/20 0.39
TAF1 P21675 1/20 0.39
BRPF1 P55201 1/20 0.39
CREBBP Q92793 1/20 0.39
CECR2 Q9BXF3 1/20 0.39
BRD9 Q9H8M2 1/20 0.39
LMNA P02545 2/20 0.37
TNF P01375 1/20 0.37
MAPT P10636 1/20 0.37
TSHR P16473 1/20 0.36
GAA P10253 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP1A2 P05177 3/20 0.35
CYP3A4 P08684 2/20 0.35
GABRA1 P14867 2/20 0.35
GABRB2 P47870 2/20 0.35
CYP11B1 P15538 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7239087 0.77 ELANE (0.41) ALDH1A1KDM4EBRD4TAF1BRPF1
SCHEMBL861748 0.73 LMNA (0.43) ALDH1A1KDM4EHTTLMNAMAPT
SCHEMBL2300077 0.69 KEAP1 (0.43) ALDH1A1KDM4EMAPTTSHRGAA
SCHEMBL2494146 0.69 ITGB3 (0.51) MAPT
SCHEMBL853110 0.68 ITGB3 (0.51) ALDH1A1KDM4EHTTMAPT
SCHEMBL2302810 0.67 TACR1 (0.41) ALDH1A1TSHRGAAL3MBTL1
SCHEMBL21615134 0.67 BRD4 (0.61) BRD4TAF1BRPF1CREBBPCECR2
SCHEMBL2301833 0.67 SLC6A2 (0.54) TSHR
SCHEMBL12380647 0.67 HSD17B10 (0.50) ALDH1A1KDM4EHTTLMNAMAPT
SCHEMBL7178642 0.67 ALDH1A1 (0.55) ALDH1A1LMNAMAPTTSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6514997-B2 Block the activity of picornaviral 3C protease AGOURON PHARMACEUTICALS, INC. 2003-02-04 US disclosed
US-20010047006-A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis AGOURON PHARMACEUTICALS, INC. 2001-11-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010047006-A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis RNASE1, SERPINB1, RNASEH1 ALDH1A1 3180/4885KDM4E 2980/4885HTT 3439/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.