SCHEMBL7296204

SCHEMBL7296204

NC(=O)[C@H](Cc1c[nH]cn1)N1CC[C@@H](Cc2ccccc2)C1=O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.43
ROCK2 O75116 1/20 0.40
ITGB2 P05107 6/20 0.38
ICAM1 P05362 6/20 0.38
ITGAL P20701 6/20 0.38
REN P00797 1/20 0.35
ALDH1A1 P00352 2/20 0.35
POLB P06746 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGAV P06756 1/20 0.35
TP53 P04637 1/20 0.35
MDM2 Q00987 1/20 0.35
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7298731 1.00 HSD11B1 (0.43) HSD11B1ROCK2ITGB2ICAM1ITGAL
SCHEMBL7295669 0.92 ROCK2 (0.41) HSD11B1ROCK2RENALDH1A1POLB
SCHEMBL7302874 0.92 ROCK2 (0.41) HSD11B1ROCK2RENALDH1A1POLB
SCHEMBL9835659 0.90 BACE1 (0.37) HSD11B1ROCK2ITGB2ICAM1ITGAL
SCHEMBL7302866 0.83 ALDH1A1 (0.36) ROCK2ITGB2ICAM1ITGALALDH1A1
SCHEMBL7294550 0.82 ALDH1A1 (0.35) ALDH1A1POLBL3MBTL1
SCHEMBL563862 0.79 HSD11B1 (0.50) HSD11B1ROCK2ITGB2ICAM1ITGAL
SCHEMBL564101 0.79 HSD11B1 (0.50) HSD11B1ROCK2ITGB2ICAM1ITGAL
SCHEMBL7291911 0.74 ALOX15 (0.37) ROCK2ALDH1A1
SCHEMBL7303150 0.73 ALDH1A1 (0.38) ALDH1A1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164388-A Hypotensive agents, treatment of congestive heart failure ABBOTT LABORATORIES (US) 1992-11-17 US disclosed
EP-0439556-A1 HETEROCYCLIC PEPTIDE RENIN INHIBITORS ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
WO-1990004917-A1 HETEROCYCLIC PEPTIDE RENIN INHIBITORS ABBOTT LABORATORIES (US) 1990-05-17 WO disclosed
EP-0365992-A1 Heterocyclic peptide renin inhibitors ABBOTT LABORATORIES (US) 1990-05-02 EP disclosed