SCHEMBL7302866

SCHEMBL7302866

NC(=O)[C@H](Cc1c[nH]cn1)N1C[C@H](Cc2ccccc2)NC1=O

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SCD O00767 1/20 0.35
ROCK2 O75116 3/20 0.35
OTUD7B Q6GQQ9 1/20 0.32
ITGB2 P05107 1/20 0.31
ICAM1 P05362 1/20 0.31
ITGAL P20701 1/20 0.31
OPRM1 P35372 2/20 0.31
OPRD1 P41143 2/20 0.31
HDAC8 Q9BY41 1/20 0.31
TP53 P04637 1/20 0.31
MDM2 Q00987 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7291911 0.92 ALOX15 (0.37) ALDH1A1SCDROCK2OTUD7B
SCHEMBL7302335 0.88 ITGB2 (0.33) ITGB2ICAM1ITGAL
SCHEMBL7294550 0.83 ALDH1A1 (0.35) ALDH1A1POLBL3MBTL1SCD
SCHEMBL7296204 0.83 HSD11B1 (0.43) ALDH1A1POLBL3MBTL1ROCK2ITGB2
SCHEMBL7298731 0.83 HSD11B1 (0.43) ALDH1A1POLBL3MBTL1ROCK2ITGB2
SCHEMBL7300912 0.82 SLC5A1 (0.31) SCD
SCHEMBL9835659 0.77 BACE1 (0.37) ALDH1A1POLBL3MBTL1ROCK2ITGB2
SCHEMBL7295669 0.74 ROCK2 (0.41) ALDH1A1POLBROCK2
SCHEMBL7302874 0.74 ROCK2 (0.41) ALDH1A1POLBROCK2
SCHEMBL7303150 0.74 ALDH1A1 (0.38) ALDH1A1POLBSCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164388-A Hypotensive agents, treatment of congestive heart failure ABBOTT LABORATORIES (US) 1992-11-17 US disclosed
EP-0439556-A1 HETEROCYCLIC PEPTIDE RENIN INHIBITORS ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
WO-1990004917-A1 HETEROCYCLIC PEPTIDE RENIN INHIBITORS ABBOTT LABORATORIES (US) 1990-05-17 WO disclosed
EP-0365992-A1 Heterocyclic peptide renin inhibitors ABBOTT LABORATORIES (US) 1990-05-02 EP disclosed