SCHEMBL7303150

SCHEMBL7303150

O=C(O)[C@H](Cc1c[nH]cn1)N1C[C@H](Cc2ccccc2)CC1=O

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
PKM P14618 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.36
ALOX15 P16050 1/20 0.36
MAPT P10636 1/20 0.36
GRM4 Q14833 1/20 0.36
SCD5 Q86SK9 2/20 0.35
SCD O00767 1/20 0.35
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
USP19 O94966 3/20 0.33
TACR3 P29371 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7294550 0.92 ALDH1A1 (0.35) ALDH1A1SMN1; SMN2GRM4SCD5SCD
SCHEMBL7291911 0.82 ALOX15 (0.37) ALDH1A1PKMSMN1; SMN2ALOX15MAPT
SCHEMBL7295669 0.81 ROCK2 (0.41) ALDH1A1PKMSMN1; SMN2ALOX15MAPT
SCHEMBL7302874 0.81 ROCK2 (0.41) ALDH1A1PKMSMN1; SMN2ALOX15MAPT
SCHEMBL9615855 0.74 BCL2 (0.46) ALDH1A1PKMALOX15POLB
SCHEMBL7302866 0.74 ALDH1A1 (0.36) ALDH1A1SCDPOLB
SCHEMBL3565608 0.74 LMNA (0.32) LMNA
SCHEMBL7296204 0.73 HSD11B1 (0.43) ALDH1A1POLBKMT2A
SCHEMBL7298731 0.73 HSD11B1 (0.43) ALDH1A1POLBKMT2A
SCHEMBL7295037 0.73 KLK7 (0.37) ALDH1A1MAPTPOLBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164388-A Hypotensive agents, treatment of congestive heart failure ABBOTT LABORATORIES (US) 1992-11-17 US disclosed
EP-0439556-A4 HETEROCYCLIC PEPTIDE RENIN INHIBITORS 1991-10-30 EP disclosed
EP-0439556-A1 HETEROCYCLIC PEPTIDE RENIN INHIBITORS ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
WO-1990004917-A1 HETEROCYCLIC PEPTIDE RENIN INHIBITORS ABBOTT LABORATORIES (US) 1990-05-17 WO disclosed
EP-0365992-A1 Heterocyclic peptide renin inhibitors ABBOTT LABORATORIES (US) 1990-05-02 EP disclosed