SCHEMBL7300368

SCHEMBL7300368

CC(C)(C)ONC(=O)CC1(Sc2ccc(Oc3ccc(F)cc3)cc2)CCOCC1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 12/20 0.40
MMP13 P45452 8/20 0.40
MMP14 P50281 5/20 0.40
MMP3 P08254 4/20 0.40
MMP9 P14780 4/20 0.40
MMP8 P22894 4/20 0.40
MMP2 P08253 3/20 0.40
MMP12 P39900 1/20 0.40
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
S1PR2 O95136 3/20 0.35
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7311858 0.91 MMP1 (0.45) MMP1MMP13MMP14MMP3MMP9
SCHEMBL7308043 0.90 MMP1 (0.46) MMP1MMP13MMP14MMP3MMP9
SCHEMBL7306527 0.88 NPC1 (0.36) MMP1MMP13MMP14MMP3MMP9
SCHEMBL7308395 0.86 MMP1 (0.48) MMP1MMP13MMP14MMP3MMP9
SCHEMBL7312678 0.82 MMP1 (0.43) MMP1MMP13MMP14MMP3MMP9
SCHEMBL7299168 0.81 LMNA (0.39) MMP1MMP13MMP2NPC1RAB9A
SCHEMBL7309991 0.80 LMNA (0.41) MMP1MMP13MMP2RAB9AALDH1A1
SCHEMBL7311907 0.79 P2RX7 (0.41) NPC1RAB9AS1PR2ALDH1A1
SCHEMBL7349344 0.78 MMP1 (0.61) MMP1MMP13MMP14MMP3MMP9
SCHEMBL7307984 0.77 ALDH1A1 (0.39) NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780386-B1 Matrix metalloprotease inhibitors HOFFMANN LA ROCHE (CH) 2002-10-02 EP disclosed
US-5932595-A ANTIARTHRITIC AGENT; MULTIPLE SCLEROSIS; OSTEOPOROSIS; RESPIRATORY SYSTEM DISORDERS; SKIN DISORDERS; ANTIULCER AGENT SYNTEX (U.S.A.) INC. (US) 1999-08-03 US disclosed
EP-0780386-A1 Matrix metalloprotease inhibitors F. HOFFMANN-LA ROCHE AG (CH) 1997-06-25 EP disclosed