SCHEMBL7307984

SCHEMBL7307984

COc1ccc(SC2(CC(=O)NOC(C)(C)C)CCCC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
NPC1 O15118 4/20 0.39
RAB9A P51151 2/20 0.39
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
TP53 P04637 1/20 0.38
AKR1B1 P15121 1/20 0.38
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
HSD11B1 P28845 1/20 0.36
EP300 Q09472 1/20 0.36
NCOA1 Q15788 1/20 0.36
NCOA3 Q9Y6Q9 1/20 0.36
EPHX2 P34913 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7299168 0.87 LMNA (0.39) ALDH1A1NPC1RAB9ALMNAPOLB
SCHEMBL7309991 0.86 LMNA (0.41) ALDH1A1RAB9ALMNAGAAMAPT
SCHEMBL7305235 0.85 MMP1 (0.47) NPC1TP53
SCHEMBL7310236 0.80 HSD11B1 (0.44) ALDH1A1NPC1MTNR1AMTNR1BTP53
SCHEMBL7311858 0.78 MMP1 (0.45) ALDH1A1LMNAGAAMAPTL3MBTL1
SCHEMBL7308043 0.77 MMP1 (0.46) ALDH1A1L3MBTL1
SCHEMBL7300368 0.77 MMP1 (0.40) ALDH1A1NPC1RAB9A
SCHEMBL7306527 0.77 NPC1 (0.36) NPC1RAB9A
SCHEMBL7304471 0.75 MMP13 (0.45)
SCHEMBL7862221 0.72 ALDH1A1 (0.61) ALDH1A1NPC1RAB9AMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780386-B1 Matrix metalloprotease inhibitors HOFFMANN LA ROCHE (CH) 2002-10-02 EP disclosed
EP-0780386-A1 Matrix metalloprotease inhibitors F. HOFFMANN-LA ROCHE AG (CH) 1997-06-25 EP disclosed